BioMAP Recommended Benchmarks

Of the over 4,500 compounds that have been profiled using the BioMAP platform, the following compounds have been curated to provide the best starting point when identifying benchmarks for your BioMAP project. Included benchmarks were selected for their complete dosing and lack of overt cytoxicity. An excel file of the table below is available for download for ease of navigation and quick filtering.
 
If you do not see a compound of interest, email us for more information about our ever expanding database.

Agent Name CAS Number Synonym Mechanism DiversityPLUS Fibrosis CRC NSCLC T Cell Panel Notes
(+/-)-Nicotine 22083-74-5 Nicotine Nicotinic Acetylcholine Receptor Agonist X
(5Z)-7-Oxozeaenol 66018-38-0 TAK1 MAPKKK Inhibitor X X
(D,L)-Mevalonic Acid Lactone 674-26-0 DL-Mevalonic Acid Lactone; Mevalonolactone HMG-CoA Reductase Inhibitor X
(R,S)-Tocopherol 10191-41-0 Vitamin E Antioxidant X
(S)-FTY720 Phosphate 402616-26-6 S1P Receptor Agonist X
(S)-Reticuline Reticuline Alkaloid X
(S)-Reticuline 3-O-sulfate CNS Depressant X
(S)-Reticuline 7-O-sulfate CNS Depressant X
15(R)-Prostaglandin D2 59894-05-2 PGD2 DP Agonist X
17α-Ethynylestradiol 57-63-6 17alpha-Ethynylestradiol ER Agonist X
17β-Estradiol 50-28-2 Estradiol ER Agonist X
1-Methyl-L-Tryptophan 21339-55-9 IDO Inhibitor X
2-(N-Ethylperfluorooctanesulfonamido)acetic Acid 2991-50-6 EtFOSAA, N-Ethylperfluorooctanesulfonamidoacetate, Et-PFOSA-AcOH Endocrine disruptor that interferes with nuclear receptor signaling and lipid metabolism X New – 2025
22(R)-Hydroxycholesterol 17954-98-2 LXRα Agonist X X
24(S)-Hydroxycholesterol 474-73-7 Cerebrosterol LXRα Agonist X
25-Hydroxyvitamin D3 19356-17-3 25(OH)D; Calcidiol; Calcifediol Vitamin D Receptor (VDR) Agonist X
2-Chloroethyl Ethyl Sulfide 693-07-2 Sulfur Mustard Vesicant X
2-Cl-IB-MECA 163042-96-4 C-Ibza-MU; Cl-IB-MECA Adenosine A3 Receptor Agonist X
2-Iodomelatonin Melatonin Receptor Agonist X
2-Methoxyestradiol 362-07-2 2-methoxy-17beta-estradiol Microtubule Disruptor X
4-Aminobenzoic Acid 150-13-0 PABA; p-Aminobenzoic Acid Vitamin B Complex Member X
5-Aminolevulinic Acid Hydrochloride Photosensitizer Precursor X
5a-POPC Cholesterol Efflux Promoter X
5-ASA 89-57-6 Apriso; Asacol; Canasa; Delzicol; Mesalazine; Mezavant; Pentasa; Rowasa; Salofalk 15-Lipoxygenase Inhibitor; COX1/2 Inhibitor; IKK1/2 Inhibitor X
5a-SM 5A-sphingomyelin Cholesterol Efflux Promoter X
666-15 1433286-70-4 CREB Inhibitor X
6-Mercaptopurine 6112-76-1 Purine Nucleotide Synthesis Inhibitor X
6-Thioguanine 154-42-7 2-Amino-6-mercaptopurine; 6-Mercaptoguanine; Thioguanine; Tioguanine Antineoplastic Agent X
8-Azaguanine 134-58-7 Azaguanine; Guanazol; Guanazolo Purine Nucleotide Synthesis Inhibitor; Xanthine Oxidase Inhibitor X
8-Br-cAMP 23583-48-4 8-Bromoadenosine; BCAMP PKA Activator X
8-CPT-cAMP 93882-12-3 Rp-Cpt-camps PKA Activator; PKG Activator X
8-Hydroxyquinoline 148-24-3 8-Quinolinol Lipophilic metal chelator X New – 2025
8-Prenylnaringenin (S)-8-dimethylallylnaringenin; 8-PN; Flavaprenin; Hopein Phytoestrogen; ER Agonist X
9-Chlorohexadecafluoro-3-oxanone-1-sulfonic Acid 73606-19-6 Potassium salt, C8 Cl-PFESA, 6:2 Chlorinated Polyfluoroalkyl Ether Sulfonate, 6:2 Chlorinated Polyfluoroalkyl Ether Sulfonic Acid, 6:2 Cl-PFAES, 6:2 Cl-PFESA, 9Cl-PF3ONS Endocrine disruptor that interferes with estrogen receptors and induces thyroid gland follicular hyperplasia. X New – 2025
9-cis-Retinoic Acid RAR/RXR Agonist X
A 205804 251992-66-2 E-selectin/ICAM-1 Inhibitor X
A23187 52665-69-7 Antibiotic A23187; Calcimycin; Ionophore A23187 Calcium Ionophore X
A939572 1032229-3-6 SCD1 Inhibitor Stearoyl-CoA Desaturase 1 Inhibitor X X
Abacavir Sulfate 188062-50-2 Abacavir; Epzicom; Ziagen Nucleoside Analog Reverse-transcriptase Inhibitor (NRTI) X
Abatacept Orencia T Cell Costimulation Modulator X
ABBV-744 2138861-99-9 BRD Inhibitor X X
Abemaciclib 1231930-82-7 LY2835219; Verzenio CDK Inhibitor X
Abiraterone 154229-19-3 CB-7598 CYP17A1 Inhibitor X
Abiraterone Acetate 154229-18-2 CB-7630; CB7630; Zytiga Cytochrome P450 17A1 Inhibitor X
Abitrexate 59-05-2 Methotrexate Tetrahydrofolate Dehydrogenase Inhbitor X
Abrocitinib 1622902-68-4 PF-04965842 JAK1 Inhibitor X
Acarbose 56180-94-0 Glucobay; Precose Maltase-glucoamylase Inhibitor; Pancreatic α-amylase Inhibitor X
ACBI1 2375564-55-7 SMARCA2, SMARCA4 and PBRM1 degrader X
ACBI2 2913161-19-8 VHL PROTAC SMARCA2 degrader X
Acebutolol Hydrochloride 34381-68-5 Sectral β1 Adrenergic Receptor Inhibitor X
Acemetacin 53164-05-9 Acemetacinum; Acemix; Emflex; Rantudil NSAID X
Acetaminophen 103-90-2 4-Acetamidophenol; APAP; Paracetamol COX-2 Inhibitor X
Acetic Acid 64-19-7 Glacial Acetic Acid Solvent X
Acetonitrile 75-05-8 Cyanomethane; Ethanenitrile; Methyl cyanide Organic Solvent X
Acitretin 55079-83-9 Ro 10-1670; Ro 10-1670/000; all-trans-Acitretin Retinoid X
Acriflavin 8048-52-0 Flavine; Panflavin Antimicrobial Agent X
Actinomycin D 50-76-0 Cosmegen; Dactinomycin RNA Polymerase Inhibitor; DNA Inhibitor X
Actinonin 13434-13-4 Actinonine; Octanohydroxamic acid Peptide Deformylase Inhibitor X
Adalimumab 331731-18-1 Humira TNFα Inhibitor X
Adapalene 106685-40-9 Adaferin; Adapaleno; Adapalenum; Differin RAR/RXR Agonist; Vitamin A Derivative; Retinoic Acid Analogue X
Adefovir Dipivoxil 142340-99-6 GS-0393; Hepsera; PMEA; Preveon Reverse Transcriptase Inhbitor X
Adenine 73-24-5 6-Aminopurine Nucleobase; Purine Derivative X
Adenosine 5-triphosphate Disodium Salt Trihydrate 34369-07-8 ATP disodium salt hydrate Metabolite X
ADU-S100 1638241-89-0 2’3’-c-di-AM(PS)2 (Rp,Rp) STING Agonist X X X
AEB071 425637-18-9 AEB-071; Sotrastaurin; UNII-7I279E1NZ8 PKCΘ Inhibitor X
AEG3482 63735-71-7 Hsp90 Inhibitor X
Afamelanotide 75921-69-6 Scenesse; melanotan-1 Melanocortin Receptor Agonist X
Afatinib 439081-18-2 BIBW2992 EGFR/HER2 Inhibitor X
AG1478 153436-53-4 AG-1478; Tyrphostin AG 1478 EGFR Inhibitor X
AIM-100 Ack1 Inhibitor X
Albendazole 54965-21-8 Albenza Microtubule Inhibitor; Anthelmintic Agent X
Aldosterone 52-39-1 Steroid hormone X New – 2025
Alectinib 1256580-46-7 Alecensa ALK Inhibitor X X X
Alemtuzumab Campath; Lemtrada Anti-CD52 Antibody X
Alendronate 121268-17-5 Fosamax Farnesyl Diphosphate Synthase Inhibitor X
Alfacalcidol 41294-56-8 1-Hydroxycholecalciferol; Bondiol; Etalpha; Oxydevit; Tevabone Vitamin D Analogue X
Alprostadil 745-65-3 Alprostadilum; Befar; Caverject; Edex; Prostaglandin E1; Prostin vr EP Agonist; Prostanoid Receptor Agonist (EP1, EP2) X
Altrenogest 850-52-2 Allyltrenbolone; Allyltrienolone; Matrix, RU-2267; Regulate Progesterone Receptor (PR) Agonist; Androgen Receptor Agonist X
Altretamine 645-05-6 Hexalen Alkylating Antineoplastic Agent X
Alverine Citrate 5560-59-8 Oxydevit; Phenpropamine Citrate Smooth Muscle Relaxant; 5-HT1A Inhibitor X
AM-966 1228690-19-4 AM966; UNII-CEO54NH393 LPA1 Receptor Inhibitor X X
AMD3465 185991-07-5 AMD 3465 Hexahydrobromide CXCR4 Inhibitor X X
Amfenac Sodium 61618-27-7 2-amino-3-benzoylbenzeneacetic Acid NSAID X
AMG208 1002304-34-8 AMG 208; UNII-Y2SR66P7VM c-Met Inhibitor X
AMG548 864249-60-5 AMG 548 p38 MAPK Inhibitor X
AMG-900 945595-80-2 Aurora Kinase Inhibitor X
Amifampridine Potassium Channel Blocker X X
Aminoglutethimide 125-84-8 Cytadren; NSC 33091 Aromatase Inhibitor X
Aminophylline 317-34-0 PDE Inhibitor; Adenosine Receptor Inhibitor X
Amitriptyline Hydrochloride 549-18-8 Elavil SNRI; TrkA Agonist; TrkB Agonist; SMase Inhibitor X
Amlexanox 68302-57-8 Amlenanox; Amoxanox; Aphthasol; Solfa Anti-inflammatory Agent; Antiallergic Agent; Immunomodulating Agent X
Amodiaquin 86-42-0 Camochin; Camoquin; Camoquine; Flavoquine Antimicrobial Agent X
Amphotericin B 1397-89-3 Abelcet; Ambisome; Amphotec Antimicrobial Agent X
Ampiroxicam 99464-64-9 NSAID X
Amprenavir 161814-49-9 Agenerase; Prozei; Vertex VX478 Protease Inhibitor X
Amylin 122384-88-7 Peptide agonist for amylin X New – 2025
Anacetrapib 875446-37-0 MK-0859 CETP Inhibitor X
Anakinra 143090-92-0 ICIL-1RA; IL-1RN; IL-1ra; IL1 Inhibitor; IRAP; Kineret IL-1 Receptor Inhibitor X
Antazoline Hydrochloride 2508-72-7 Vasocon-a H1 Receptor Inhibitor X
Antimycin A 1397-94-0 Antimycin A1; Antimycin A1b; Antipiricullin; Fintrol; Virosin Cytochrome c Reductase Inhibitor; Mitochondrial Inhibitor X
Apelin-13 Apelin Receptor (APJ) Ligand X
Apoptolidin 194874-06-1 Apoptosis Activator IV; Nocardiopsis sp. F(0)F(1) ATPase Inhibitor; Mitochondrial Inhibitor X
Apremilast 608141-41-9; Apremilastum; CC 10004; CC-10004; Otezla PDE4 Inhibitor X
APX-3330 136164-66-4 Erenapurstat; E3330 Inhibitor of Ape-1/Ref-1 redox X New – 2025
Artemisinin 63968-64-9 NSC 369397 Antimicrobial Agent X
Articaine Hydrochloride 23964-57-0 Carticaine Anesthetic Agent X
ARV-825 1818885-28-7 BRD4 PROTAC X
AS1892802 928320-12-1 AS 1892802; AS-1892802 ROCK1, ROCK2 Inhibitor X
AS2444697 AKOS027470180 IRAK4 Inhibitor X
AS601245 345987-15-7 AS 601245 JNK Inhibitor X
AS605240 648450-29-7 PI 3-Kgamma Inhibitor; PI3-Kγ Inhibitor PI3K Inhibitor X
Asciminib 1492952-76-7 ABL001 BCR-ABL1 inhibitor X
Asenapine 85650-56-2 Antipsychotic Agent X
Aspirin 50-78-2 Acetylsalicylate; Acetylsalicylic acid COX Inhibitor X
Astemizole 68844-77-9 Astemison; Astemizol; Astemizolum Antihistamine Agent X
Atazanavir Sulfate 229975-97-7 BMS 232632; CGP 73547; Reyataz HIV Protease Inhibitor X
Atlizumab 375823-41-9 Actemra; MRA; RoActemra; Tocilizumab IL-6 Receptor Inhibitor X
Atomoxetine Hydrochloride 82248-59-7 Strattera Norepinephrine Reuptake Inhibitor X
Atorvastatin 134523-00-5 Lipitor; Lipovastatinklonal HMG-CoA Reductase Inhibitor X
Atovaquone 95233-18-4 Atavaquone Cytochrome b Inhibitor X
ATP Adenosine triphosphate Coenzyme X
Atracurium Besylate 64228-81-5 64228-81-5; Atracurium Besilate; Atracurium Besylate; Tracrium Neuromuscular Blocking Agent X
Auranofin 34031-32-8 NSC 321521; Ridauragold thiol; SKF 39162 Thioredoxin Reductase Inhibitor X
Avacopan 1346623-17-3 CCX168 Complement 5a receptor Inhibitor X
AVL-292 CC-292; Spebrutinib BTK Inhibitor X X X
AX-15836 2035509-96-5 ERK5 Inhibitor X
Axitinib 319460-85-0 Inlyta VEGFR2 Inhibitor X X X X
AZ876 898800-26-5 LPM029_300383_00 LXR Agonist X
Azaperone 1649-18-9 R-1929; Stresnil; Suicalm Dopamine Receptor Inhibitor X
Azatadine Dimaleate 3978-86-7 Azatadine Maleate; Bonamid; Idulian Histamine and Cholinergic Inhibitor X
Azathioprine 446-86-6 Azasan; BW-57-322; Imuran Purine Metabolism Anatgonist X X
AZD1208 1204144-28-4 AZD 1208 PIM Kinase Inhibitor X
AZD4547 1035270-39-3 AZD 4547; AZD-4547 FGFR Inhibitor X
AZD8055 1009298-09-2 AZD 8055; AZD-8055 mTOR Inhibitor X
Azithromycin 83905-01-5 Azasite; Azenil; Azifast; Azigram; Azimakrol; Hemomycin; Zithromax Antibiotic Agent X X
Bacitracin Zinc 1405-89-6 Antibiotic Agent X
Bafilomycin A1 88899-55-2 NSC 381866 V-ATPase Inhibitor X
Baricitinib 1187594-09-7 INCB 028050; LY3009104 JAK1/2 Inhibitor X
BAY 2666605 2275774-60-0 PDE3A/B Inhibitor X
BAY-876 1799753-84-6 GLUT1 Inhibitor X
BBO-8520 2893809-51-1 Inhibitor targeting KRAS X New – 2025
BDH35145960b BET Inhibitor X
BDV0005266b Bromodomain Inhibitor X
Beclomethasone Dipropionate 4419-39-0 Qvar GR Agonist X
Bedaquiline EX00040046; Sirturo Mycobacterial ATP Synthase Inhibitor X
Belatacept T Cell Costimulation Modulator X
Belimumab Benlysta BAFF Inhibitor X
Belinostat 866323-14-0 PXD101; PX105684 HDAC Inhibitor X
Belumosudil 911417-87-3 KD025 synonym selective inhibitor of ROCK2 X New – 2025
Bemcentinib 1037624-75-1 BGB324; R428 AXL Inhibitor X X X X
Benzethonium Chloride 121-54-0 Antiseptol; BZT; Diapp; Disilyn; Hyamine; Phemithyn; Phermerol; Polymine D; Quatrachlor; Salanine Antimicrobial Agent; AChE Inhibitor X
Benzocaine 94-09-7 Americaine; Ethyl Aminobenzoate Anesthetic X
Benztropine Mesylate 132-17-2 Cogentin Muscarinic Acetylcholine Receptor (mAChR) Inhibitor X
Benzydamine Hydrochloride 132-69-4 AF-864; Tantum NSAID X
Beraprost MDL-201229; Procylin Prostacyclin Analogue X
Berberine Berberin; Umbellatine Dipeptidyl Peptidase IV Inhibitor; PTP1B Inhibitor X
Bergapten 484-20-8 5-Methoxypsoralen; Bergaptene; Heraclin; Majudi Psoralen X
beta-Mercaptoethanol Inorganic Compound X X
Betamethasone 378-44-9 Celestone Glucocorticoid Receptor (GR) Agonist X
Betamethasone Dipropionate 5593-20-4 Diprolene Glucocorticoid Receptor (GR) Agonist X
Betamethasone Valerate 2152-44-5 Betnovate Glucocorticoid Receptor (GR) Agonist X
Betamipron 3440-28-6 Benzoyl-beta-alanine Carbapenem Antibiotic Agent X
Betapar 1247-42-3 Betanisona; Meprednisone; Methylprednisone Glucocorticoid Receptor (GR) Agonist X
Bevacizumab 216974-75-3 Avastin; anti-VEGF VEGFA Inhibitor X X
Bexagliflozin 1118567-05-7 EGT-1442, THR-1442 Potent and selective SGLT2 inhibitor X New – 2025
BI-10n ITK Inhibitor X
BI2536 755038-02-9 BET Inhibitor; PLK1 Inhibitor X X
BI-2545 2162961-71-7 Autotaxin Inhibitor X X X X
BI-3663 2341740-84-7 PTK2/FAK PROTAC X
BI-7273 1883429-21-7 BRD7/9 Inhibitor X
BIBX1382 196612-93-8 BIBX 1382; Falnidamol EGFR Inhibitor X
Bilirubin 635-65-4 Bilirubin IX- α; Hematoidin; Hemetoidin Heme Metabolite X
Bindarit CCL2/7/8 Inhibitor X
Biperiden Hydrochloride 1235-82-1 Akineton; Akinophyl Acetylcholine Inhibitor X
Bisacodyl 603-50-9 Bicol; Brocalax; Dulcolax; Durolax Laxative X
Bismuth Subcitrate Potassium 880149-29-1 Bismuth Subcitrate; Bismuth Subcitrate Potassium; De-Noltab; Gastrodenol; Tripotassium Dicitratobismuthate Antibiotic Agent X
Bisphenol A 80-05-7 Endocrine-disrupting toxicant X New – 2025
Bleomycin Sulfate 9041-93-4 Blenoxane; Bleomycin Antineoplastic Agent X
BMP7 Osteogenic Protein-1 (OP-1) Activin Receptor Agonist (Activin RIA, RIIA, RIIB; BMPR-IA, BMPR-IB, BMPR-II) X
BMS-777607 1025720-94-8 BMS777607 c-Met Inhibitor; Axl Inhibitor; RON Inhibitor; Tyro3 Inhibitor X X X
BMS-986365 2446928-30-7 CC-94676 Androgen receptor (AR) PROTAC degrader. X New – 2025
BMY 45778 152575-66-1 Non-prostanoid Prostacyclin IP Receptor Partial Agonist. X
Bortezomib 179324-69-7 Velcade Proteasome Inhibitor X X
Bosentan 147536-97-8 Bosentan Hydrate; Bosentanum; Tracleer ET-A Inhibitor; ET-B Inhibitor X
Bosutinib 380843-75-4 Bosulif; SKI-606 BCR-ABL Inhibitor; Src Inhibitor X X X
Branaplam 1562338-42-4 LMI070; NVS-SM1 survival motor neuron-2 splicing modulator X New – 2025
Brefeldin A 20350-15-6 Ascotoxin; Cyanein; Decumbin; Synergisidin ARF1 Inhibitor X
Brequinar Bay_BioMAP_005_B2; bipenquinate DHODH Inhibitor X
Brigatinib ALK Inhibitor; EGFR Inhibitor X X
Bromfenac Sodium 91714-93-1 Xibrom NSAID; COX Inhibitor X
Bromosporine 1619994-69-2 Pan Bromo Domain Inhibitor X
Brompheniramine Maleate 980-71-2 BPN; Bromfed; Bromfenex; Dimetane; Dimetapp; Lodrane Antihistamine Agent X
Broxyquinoline 521-74-4 Dibromohydroxyquinoline Antimicrobial Agent X
BSK_4925 Not Listed Lymphocyte Specific Kinase Lck Inhibitor X
BSK_anti-CTLA4 Not Listed CTLA4 Inhibitor X
Bucladesine 362-74-3 Actosin; Dibutyryl cAMP; Dibutyryl cyclic AMP PDE4 Inhibitor X
Budesonide 51333-22-3 Budeson; Entocort; Preferid; Pulmicort; Spirocort Glucocorticoid Receptor (GR) Agonist X X X
Bupropion Hydrochloride 34841-39-9 Amfebutamone; Budeprion; Bupropion; Elontril; Prexaton; Quomem; Voxra; Wellbutrin NDRI X
Busulfan 55-98-1 Busulfex; Myleran Alkylating Antineoplastic Agent X
BW 245C 75693-75-3 BW-245C; BW245C DP Agonist X
BW 246C 65705-83-1 8-epi BW 245C DP Agonist X
C188-9 432001-19-9 TTI-101 STAT3 Inhibitor X X
Cabozantinib 849217-68-1 BMS-907351; Cometriq; XL184 VEGFR2 Inhibitor X X X X
Caffeine 58-08-2 1,3,7-Trimethylxanthine, Caffeine Agonist of Adenosine receptor X New – 2025
Calcipotriene 112965-21-6 Daivonex; Dovonex; Sorilux Synthetic Calcitriol Derivative X
Calcitriol 32222-06-3 Calcijex; Calcitriolum; Decostriol; Rocaltrol; Silkis; Vectical Vitamin D Receptor (VDR) Agonist X
Calcium Chloride 10043-52-4 CaCl2; Calcium Chloride Anhydrous Salt X
Camostat Mesylate 59721-29-8 FOY305; FOY0S980 Serine Protease Inhibitor X X
Canakinumab 914613-48-2 Ilaris; ACZ885, ACZ-885 IL-1β Sink X
Cantharidin 56-25-7 Cantharone Protein Phosphatase 2A (PP2A) Inhibitor X
CAPE 104594-70-9 Caffeic Acid Phenethyl Ester; Phenethyl caffeate 15-Lipoxygenase Inhibitor X
Carbimazole 22232-54-8 Athyromazole Antithyroid Agent X
Carboplatin Paraplat; Paraplatin; Paraplatin-AQ DNA Repair Inhibitor X
Carfilzomib 868540-17-4 Kyprolis; PR-171 Proteasome Inhibitor X
Carmofur 61422-45-5 1-hexylcarbamoyl-5-fluorouracil; HCFU Pyrimidine Analogue; Antineoplastic Agent X
Carprofen 53716-49-7 Imadyl; Imafen; Novox; Quellin; Rimadyl; Rovera; Vetprofen NSAID X
Carvedilol 72956-09-3 Beta Blocker; Carvedilolum; Coreg; Coreg CR; SKF 105517 Adrenergic Receptor Inhibitor X
Caspofungin Acetate 179463-17-3 Cancidas; L-743,872; MK 0991 Antimicrobial Agent X
CAY10410 596104-94-8 9,10-dihydro-15-deoxy-Δ12,14-PGJ2 PPARγ Agonist X
CCG-1423 285986-88-1 Myocardin-related Transcription Factor-A MRTF-A Inhibitor; Rho Kinase/ROCK Signaling Inhibitor X X
CDDO Methyl Ester 218600-53-4 Bardoxolone Methyl; NSC 713200; RTA 402; TP-155 Nrf2 Activator; Triterpenes X
Ceftazidime Pentahydrate 78439-06-2 Fortaz; Tazicef Antibiotic Agent X
Celecoxib 169590-42-5 Celebrex, Celecoxibum COX-2 Inhibitor X New – 2025
Cepharanthine 481-49-2 Anti-inflammatory Agent; Antineoplastic Agent X
Cerivastatin 143201-11-0 Baycol; Cerivastatin Acid; Lipobay HMG-CoA Reductase Inhibitor X
Cetirizine Dihydrochloride 83881-51-0 Alerlisin; Reactine; Zyrtec Antihistamine Agent; GPCR Ligand X
Cetrimonium Bromide 57-09-0 CTAB; Centimide; Cetyltrimethylammonium Bromide; Hexadecyltrimethylammonium Bromide Antimicrobial Agent X
Cetuximab Anti-EGFR; Erbitux; IMC-C225 EGFR Inhibitor X X X
Cetylpyridinium Chloride 123-03-5 Antiseptic Agent X
CFM 1571 Hydrochloride sGC Activator X
CGP 52608 87958-67-6 RORα Ligand X
CH223191 301326-22-7 AhR Inhibitor X
CHIR-99021 Hydrochloride 252917-06-9 CT99021 GSK-3α/β Inhibitor X X
Chlorambucil 305-03-3 Ambochlorin; CHLORAMBUCIL; Chloraminophen; Leukeran Alkylating Agent X
Chlorocresol 59-50-7 4-chloro-3-cresol; 4-chloro-3-methylphenol Antiseptic Agent X
Chloroquine Phosphate 50-63-5 Aralen; Resoquine; Reumachlor; Sanoquin Antimicrobial Agent X
Chlorothiazide 58-94-6 Diuril Antihypertensive Agent; Diuretic Agent X
Chlorprothixene 113-59-7 Chlorprothixenum; Clorprotixeno; Taractan; Truxal Antipsychotic Agent X
Chlorquinaldol 72-80-0 Sterosan Antimicrobial Agent X
Cholecalciferol 67-97-0 Calciol; Colecalciferol; Oleovitamin D3; Vitamin D3 Vitamin D Receptor (VDR) Agonist X
Cilnidipine 132203-70-4 Atelec; Cinalong; Siscard Calcium Channel Blocker X
Cilostazol 73963-72-1 Cilostazole; Cilostazolum; Pletaal; Pletal PDE Inhibitor XZ
Cinacalcet Hydrochloride 364782-34-3 AMG-073 HCl Calcimimetic Agent; Extracellular Calcium-sensing Receptor Agonist X
Cinchophen 132-60-5 Atophan; Phenaquin; Quinophan Analgesic Drug X
Ciprofloxacin Hydrochloride 85721-33-1 BAY-o 9867; Cetraxal; Ciloxan; Cipro; Ciprol; NSC 620634 Antimicrobial Agent X
Cisplatin 15663-27-1 CACP; Cisplatina; Cisplatinum; DDP; Neoplatin; Platinol-AQ DNA Alkylating Agent X X
Cladribine 4291-63-8 2-CdA; 2-Chlorodeoxyadenosine; Leustatin Antineoplastic Agent X
Clemastine 17-7-4 Clemastina; Clemastinum Antihistamine Agent X
Clexane Ardeparin; Enoxaparin; Enoxaparin Sodium; Heparin; Nadroparin; Tinzaparin Anticoagulant Agent X
CLI-095 Meclastin; Resatorvid; TAK-242 TLR4 Inhibitor X X X
Climbazole 38083-17-9 Baypival; Baysan Antimicrobial Agent X
Clofarabine 123318-82-1 CAFdA; Clofarex; Clolar; Evoltra Nucleic Acid Synthesis Inhibitor X
Clofazimine 2030-63-9 Lamprene Antimycobacterial Agent X
Cloprostenol (+)-16-m-chlorophenoxy Tetranor Prostaglandin F2α Prostaglandin F (FP) Receptor Agonist; PGF2α Analog X
Closantel Sodium 61438-64-0 Antimicrobial Agent X
Clozapine 5786-21-0 Clozapinum; Clozaril; Fazaclo; Versacloz Antipsychotic Agent X
Cobalt(II) Chloride Hexahydrate 7791-13-1 Cobaltous Chloride Hexahydrate Inorganic Compound X X
Cobicistat 1004316-88-4 GS-9350; GS-9350, Tybost; Tybost CYP3A Inhibitor
Coffee Extract Coffee Extract X
COH34 906439-72-3 PARG inhibitor X New – 2025
Colchicine 114977-28-5 Colchicin; Colchicina; Colchicinum; Colcrys; Mitigare Microtubule Disruptor X X X
Concanamycin A 80890-47-7 Antibiotic X 4357B; NSC 674620; X 4357B V-ATPase Inhibitor X
Concanavalin A Type VI 11028-71-0 Purified Lectin X
Copper(II) Sulfate 7758-98-7 Glucose-6-phosphate Dehydrogenase (G6PD) Inhibitor; Paraoxonase Inhibitor X
Cortistatin-14 186901-48-4 Cortistatin14 Steroidal Alkaloids X
CP 55,940 Cannabinoid (CB) Receptor Agonist X
CPG 52364 TLR7/TLR8/TLR9 Inhibitor X
Crisaborole Eucrisa PDE4 Inhibitor X
Crizotinib 877399-52-5 PF 2341066; PF-02341066; Xalkori Anticancer Agent; ALK Tyrosine Kinase Receptor Inhibitor; HGFR Inhibitor X X X
Cudetaxestat 1782070-21-6 BLD-0409, PAT-409 ATX Inhibitor X New – 2025
Curcumin Natural Phenol X X X
Cyanocobalamin 68-19-9 Cyanocob(III)alamin; Nascobal; Vitamin B12 Vitamin B12 Analogue X
Cycloheximide 66-81-9 Actidione; Cicloheximide; Kaken; Naramycin A Protein Synthesis Inhibitor X
Cyclopentyl Adenosine Adenosine A1 Receptor Agonist X
Cyclosporin A 59865-13-3 CyA; Cyclosporine; Gengraf; Neoral; Restasis; Sandimmune Calcineurin Inhibitor; Cyclophilin A Modulator X X X X
Cystamine dihydrochloride 56-17-7 Transglutaminase inhibitor X New – 2025
Cysteamine hydrochloride 156-57-0 2-Aminoethanethiol hydrochloride 2-Aminoethanethiol hydrochloride; 2-Mercaptoethylamine hydrochloride X New – 2025
Cytarabine 147-94-4 Ara-C; Arabinosylcytosine; Cytosar; Cytosine Arabinoside DNA Synthesis Inhibitor X
Dabrafenib GSK2118436; Tafinlar BRAF Inhibitor X X X
Dacomitinib Vizimpro EGFR Inhibitor X X
Dactolisib 915019-65-7 BEZ235; NVP-BEZ235 PI3K Inhibitor; mTOR Inhibitor X X X
Dalcetrapib 211513-37-0 JTT-705 Cholesterylester Transfer Protein (CETP) Inhibitor X
Danofloxacin Mesylate 119478-55-6 Advoci; CP-76136-27; Nofloxacin Antimicrobial Agent X
Danusertib 827318-97-8 PHA-739358 Aurora Kinase Inhibitor X
Daprodustat 960539-70-2 GSK1278863 Hypoxia-inducible factor-prolyl hydroxylase (HIF-PH) inhibitor X New – 2025
Daratumumab 945721-28-8 Anti-Human CD38, Human Antibody Anti-CD38 Antibody X
Darifenacin Hydrogen Bromide 133099-07-7 Enablex; UK 88525-04 Muscarinic Acetylcholine Receptor Inhibitor X
Darunavir Ethanolate 635728-49-3 Prezista; TMC114 Protease Inhibitor X
Dasatinib 302962-49-8 BMS-354825; Sprycel Multikinase Inhibitor (Src tyr Kinase, BCR/Abl) X X X X
Daunorubicin Hydrochloride 23541-50-6 Acetyladriamycin; Daunomycin; Daunorubicina; Daunorubicine ; Daunorubicinum; Leukaemomycin C; Rubidomycin DNA Topoisomerase Inhibitor X X
dBET1 1799711-21-9 BRD4 PROTAC X
Decitabine 2353-33-5 Azadc; Dacogen; Dezocitidine Nucleic Acid Synthesis Inhibitor X
Defactinib 1073154-85-4 VS-6063; PF-04554878 FAK inhibitor X New – 2025
Defactinib 1073154-85-4 VS-6063; PF-04554878 FAK inhibitor X New – 2025
Deferasirox 201530-41-8 Exjade; ICL670A Iron Chelating Agent X
Deferoxamine Mesylate 70-51-9 DFOA; DFOM; Deferoxamina; Deferoxamine; Deferoxaminum; Deferrioxamine Iron Chelating Agent X
Denosumab Prolia; Xgeva RANKL Inhibitor X X
Deoxyarbutin 53936-56-4 Tyrosinase Inhibitor X
Dequalinium Chloride 522-51-0 Danical; Decabis; Dequafungan Antimicrobial Agent; PKC Inhibitor X
Deruxtecan 1599440-13-7 MC-GGFG-DXD ADC Payload X
Desloratadine 100643-71-8 Aerius; Clarinex; Descarboethoxyloratadine Antihistamine Agent X
Desonide 638-94-8 Desowen; Tridesilon Glucocorticoid Receptor (GR) Agonist X
Deucravacitinib 1609392-27-9 BMS-986165 Tyk2 Inhibitor X X
Dexamethasone 50-02-2 Baycadron; Decadron; Dexametasona; Maxidex; Ozurdex Glucocorticoid Receptor (GR) Agonist X X X
Dexlansoprazole 138530-94-6 Dexilant; Kapidex Proton Pump Inhibitor X
Dexmedetomidine 113775-47-6 Dex; Precedex α2 Adrenergic Receptor Agonist X
Dextromethorphan 125-71-3 DXM, D-Methorphan Noncompetitive NMDA receptor antagonist X New – 2025
Dibucaine 85-79-0 Cinchocaine; Dermacaine; Nupercainal; Nupercaine Anesthetic X
Diclofenac Diethylamine 78213-16-8 AK163134; UNII-6TGQ35Z71K NSAID X
Diclofenac Potassium 15307-81-0 Cambia; Cataflam; UNII-L4D5UA6CB4; Zipsor NSAID X
Dienogest 65928-58-7 Progestin; Visanne Semisynthetic Steroidal Progestogen X
Diethylstilbestrol 56-53-1 11β-hydroxysteroid dehydrogenase 2 inhibitor X New – 2025
Difluprednate 23674-86-4 Durezol Corticosteroid X
Digoxigenin 1672-46-4 Digitoxigenin; Uzarigenin Hapten X
Dihydrotestosterone 521-18-6 Anaboleen; Androlone; Androstanolone; Stanaprol; Stanolone AR Agonist X
Dimethyl Fumarate 624-49-7 BG-12; DMF; Tecifidera NFκB Inhibitor; Nrf2 Activator X
Diminazene Aceturate 908-54-3 Diminazeno; Diminazenum ACE Activator X
Diphenylpyraline Hydrochloride 132-18-3 Allerzine; Diaphen; Histalert Antihistamine Agent; GPCR Ligand X
Diprophylline 479-18-5 Dilor PDE Inhibitor; Adenosine Receptor Antagonist X
Dipyridamole 58-32-2 Cardoxin; Cleridium 150; Curantyl; Permole; Persantin; Persantine PDE Inhibitor X X
Disulfiram 97-77-8 Antabuse; Tetraethylthiuram Disulfide Aldehyde Dehydrogenase Inhibitor X
Donepezil Hydrochloride 120011-70-3 Aricept; Donepezilum Cholinesterase Inhibitor X
Doramapimod 285983-48-4 BIRB-796; BIRB796 p38 MAPK Inhibitor X X
Dorzolamide Hydrochloride 120279-96-1 MK-507 Carbonic Anhydrase Inhibitor X
Doxazosin Mesylate 74191-85-8 Cardura α1 Adrenergic Receptor Inhibitor X
Doxorubicin Hydrochloride 25316-40-9 Adriamycin; Doxorubicine; Doxorubicinum; Hydroxydaunorubicin DNA Topoisomerase Inhibitor X
D-Pantethine 16816-67-4 Pantethine; Pantetina; Pantomin; Pantosin Cofactor Precursor X
Droperidol 548-73-2 Dehydrobenzperidol; Dridol; Droleptan; Inapsine Dopamine Receptor (D2) Inhibitor; 5-HT2A Receptor Inhibitor X
Drospirenone 67392-87-4 1,2-dihydrospirorenone; Yasmin Progesterone Receptor (PR) Agonist X
Dupilumab 1190264-60-8 REGN-668 Anti-IL-4 Antibody X X
Durvalumab Imfinzi Anti-PD-L1 Antibody X X
Dydrogesterone 152-62-5 Duphaston; Isopregnenone Progesterone Receptor (PR) Agonist X
Edaravone 89-25-8 MCI-186; Radicut Antioxidant X
Eflornithine 70052-12-9 DFMO; MDL71782; RMI71782; α-difluoromethylornithine Ornithine Decarboxylase Inhibitor X
EGF 62253-63-8 Epidermal Growth Factor EGFR Activator X
EGFR/ErbB-2/ErbB-4 Inhibitor 881001-19-0 EGFR Inhibitor; HER2, HER4 Inhibitor X
Eicosapentaenoic Acid 10417-94-4 EPA; Icosapentaenoic Acid Omega-3 Fatty Acid; Eicosanoid Precursor X
Elafibranor 923978-27-2 GFT505 PPARα/δ agonist X X
Elesclomol 488832-69-5 STA-4783 ROS Inducer X
Ellagic Acid 476-66-4 Antioxidant Agent X
Embelin X-linked Inhibitor of Apoptosis Protein (XIAP) Inhibitor X
Emricasan 254750-02-2 Caspase Inhibitor X
Enbrel 185243-69-0 Etanercept; TNF-R2 TNFα Inhibitor X
ENMD-2076 934353-76-1 Kinase Inhibitor X
Entinostat 209783-80-2 MS-275; SNDX-275 HDAC Inhibitor X
Entrectinib 1108743-60-7 NMS-E628 TrkA/B/C/ROS1/ALK Inhibitor X X X
Epacadostat INCB024360 IDO Inhibitor X X X
Epalrestat 82159-09-9 ONO-2235 Aldose Reductase Inhibitor X X
Epothilone B 152044-54-7 EPO 906; EPO906; Patupilone Microtubule Disruptor X
Epothilone D 189453-10-9 Desoxyepothilone B Microtubule Disruptor X X X
Eprazinone Dihydrochloride 10402-53-6 746CE; Eftapan; Mucitux; NSC 317935; Resplen; Rozuplen Mucolytic Agent X
Eribulin Mesylate 441045-17-6 E7389 Microtubule Binder X X X
ERK5-IN-1 1234479-76-5 ERK5 Inhibitor X
Erlotinib 183321-74-6 CP-358,774; Erlotinib Hydrochloride; OSI-774; Tarceva EGFR Inhibitor X X X X
Erythromycin 114-07-8 Abomacetin; Eritromicina; Ilotycin Antibiotic Agent X
Ethacridine Lactate 6402-23-9 Acrinol; Rivanol DNA Intercalating Antiseptic Agent X
Ethacrynic Acid 58-54-8 Edecrin Diuretic Agent X
Ethanol 64-17-5 Alcohol; Ethyl Alcohol; Ethyl Hydroxide GABA-A Receptor Agonist; NMDA Receptor Inhibitor X
Ethionamide 536-33-4 Antimicrobial Agent X
Ethosuximide 77-67-8 Aethosuximide; Atysmal; Ethosuximidum; Etosuximida Voltage-gated T-type Calcium Channel Blocker X
Ethoxzolamide 452-35-7 Ethoxyzolamide Carbonic Anhydrase Inhibitor X
Ethyl Pyruvate 617-35-6 Ethyl 2-Oxopropanoate; Pyruvic Acid Ethyl Ester Anti-inflammatory Agent X
Ethylenediamine 107-15-3 Organic Compound X
Etodolac 41340-25-4 Etodolaco; Etodolacum; Etodolic acid; Lodine COX-2 Inhibitor X
Etomidate 33125-97-2 Amidate Anaesthetic Agent; GABA-A Agonist X
Etoposide 33419-42-0 VP-16 DNA Topoisomerase (TOPO) II Inhibitor X
Etrasimod 1206123-37-6 APD334 S1P receptor modulator X New – 2025
Etravirine 269055-15-4 Intelence; TMC-125; TMC125 NNRTI X
Everolimus 159351-69-6 Afinitor; Certican; Evertor; RAD001; Zortress mTOR Inhibitor X X X X
Exemestane 107868-30-4 Aromasin Steroidal Aromatase Inhibitor X
Ezetimibe 163222-33-1 Ezedoc; SCH-58235; Zetia Antilipemic Agent X
Famprofazone 22881-35-2 Gewodin; Gewolen NSAID X
Fasudil 103745-39-7 Fasudil Hydrochloride; HA-1077 ROCK1, ROCK2 Inhibitor X X
FCCP 370-86-5 Carbonyl cyanide p-trifluoromethoxyphenylhydrazone Uncoupling Agent; Ionophore X
Febuxostat 144060-53-7 Adenuric; Feburic; Goturic; Uloric Xanthine Oxidase Inhibitor X
Fedratinib 936091-26-8 Inrebic; SAR302503; TG101348 JAK2 Inhibitor X X
Fenbendazole 43210-67-9 Panacur Anthelmintic Agent; Microtubule Disruptor X
Fenoprofen Calcium Dihydrate 34597-40-5 Fenopron; Nalgesic; Progesic COX Inhibitor X
Fenspiride Hydrochloride NAT-333; NDR-5998A PDE Inhibitor X
Fexofenadine Hydrochloride 153439-40-8 Allegra H1 Receptor Inhibitor X
Fezolinetant 1629229-37-3 ESN-364 neurokinin 3 receptor antagonist X New – 2025
FICZ 172922-91-7 AhR Agonist X X
Fidaxomicin 873857-62-6 Dificid; Dificlir; OPT-80; PAR-101 Antibiotic Agent X
Filgotinib GLPG0634 JAK1 Inhibitor X X X
Finasteride 98319-26-7 Propecia; Proscar Type II, Type III 5α-reductase Inhibitor X
Fingolimod 162359-56-0 FTY720; Gilenya S1P Receptor Agonist X
Flagellin TLR5 Agonist X
Fleroxacin 79660-72-3 FLRX; Megalone ; Megalosin; Quinodis Antimicrobial Agent X
Flubendazole 31430-15-6 Flutelmium Antimicrobial Agent X
Fludarabine 21679-14-1 2-Fluoro-Ara-A; F-ara-A; Fludara; NSC 118218; Oforta STAT1 Inhibitor; DNA Synthesis Inhibitor X
Fludrocortisone 127-31-1 Fludrocortisona; Fludrocortisonum; Fluohydrocortisone Glucocorticoid Receptor (GR) Agonist; Mineralocorticoid Receptor (MR Agonist) X
Flumazenil 78755-81-4 Anexate; Flumazepil; Lanexat GABA/Benzodiazepine Receptor Inhibitor X
Flumethasone 2002-29-1 Locacorten; Locorten; Orsalin; U-10974 Glucocorticoid Receptor (GR) Agonist X
Flunarizine Dihydrochloride 30484-77-6 Flunarizina Calcium Channel Blocker; Antihistamine Agent X
Fluorometholone Acetate Eflone; Flarex; Fluorometholone 17-acetate; Oxylone Acetate Glucocorticoid Receptor (GR) Agonist X
Fluorouracil 51-21-8 5-FU; 5-FU; 5-Fluracil; Adrucil; Fluoro Uracil; Fluoroplex; Fluouracil Thymidylate Synthase (TS) Inhibitor; Pyrimidine Analog X X
Fluoxetine 54910-89-3 Adofen; LY-110140; Prozac; Sarafem; Symbyax Antidepressant; SSRI Inhibitor X
Flurbiprofen 5104-49-4 Ansaid; FLP; Ocufen COX Inhibitor; NSAID X
Fluticasone Propionate 80474-14-2 Fluticason; Fluticasona; Fluticasone; Fluticasonum Glucocorticoid Receptor (GR) Agonist; Progesterone Receptor (PR) Agonist X X
Fluvastatin 93957-54-1 Fluvastatin Sodium; Lescol HMG-CoA Reductase Inhibitor X
Fluvoxamine Maleate 61718-82-9 Luvox SSRI X
FM-381 DRX_FM-381 JAK3 Inhibitor X
fMLP 59880-97-6 FMLP; N-Formylmethionyl-leucyl-phenylalanine FPR Agonist X
Forskolin 66575-29-9 Coleonol; Colforsin; Colforsina; Colforsine Adenylyl Cyclase Activator X
Fosaprepitant Dimeglumine 265121-04-8 Ivemend; L 758298; UNII-6L8OF9XRDC Neurokinin-1 Receptor Inhibitor X
Fosbretabulin Disodium 168555-66-6 CA4DP; Zybrestat Microtubule Disruptor X
Foscenvivint 1422253-38-0 PRI-724 CBP/β-Catenin Inhibitor X
Fostamatinib 1025687-58-4 R406 Syk Inhibitor X
FR180204 865362-74-9 ERK Inhibitor X
FSL-1 TLR2/TLR6 Agonist X
Ftorafur 17902-23-7 Tefudex; Tegafur-uracil; UFT; Uftotral; Ufur Chemotherapeutic Agent X
Fucoidan 9072-19-9 Caspase-3 Activator X
Fulvestrant 129453-61-8 Faslodex Estrogen Receptor (ER) Inhibitor X
Fumagillin 23110-15-8 Fumidil Angiogenesis Inhibitor; MetAP2 Inhibitor X
Galeterone 851983-85-2 TOK-001 CYP17A1 Inhibitor X
Galunisertib 700874-72-2 LY2157299 TGFβR1 Kinase Inhibitor X X X X
Gandotinib 1229236-86-5 LY2784544 JAK2 Inhibitor X X
GB1107 1978336-61-6 Inhibitor of Galectin-3 X New – 2025
GDC0834 1133432-49-1 BTK Inhibitor X X X
GDC0853 RG-7845 BTK Inhibitor X
GDC0879 B-Raf/C-Raf Inhibitor X
GDC0941 957054-30-7 GDC-0941; Pictilisib PI3Kα/δ Inhibitor X X X X
Gefitinib 184475-35-2 Iressa; ZD 1839 EGFR Inhibitor X X
Geldanamycin 30562-34-6 Geldanomycin Hsp90 Inhibitor X X
Gemcitabine Hydrochloride 122111-03-9 Gemzar; LY-188011; dFdC; dFdCyd Nucleoside Metabolic Inhibitor  X X X
Gemfibrozil 25812-30-0 Gemfibrozilo; Gemfibrozilum; Lopid PPARα Agonist X
Genistein 446-72-0 Genisteol; Genisterin; NSC-36586 Phytoestrogen X
Gestodene 60282-87-3 15-dehydronorgestrel Progesterone Receptor (PR) Agonist X
GF109203X 133052-90-1 Bisindolylmaleimide I PKC (c+n) Inhibitor X
Gilteritinib 1254053-43-4 Xospata Tyrosine Kinase Inhibitor X
GKT137831 1218942-37-0 GKT-137831 NOX1/NOX4 Inhibitor X X
Glasdegib 1095173-27-5 PF-04449913 Smoothened (SMO) Inhibitor X
Glatimer Acetate Copaxone Immunomodulating Agent X
Glesatinib Tyrosine Kinase Inhibitor X
Gliquidone 33342-05-1 Beglynor; Glikvidon; Gliquidonum; Glurenorm KATP Channel Blocker X
GLP-1 Proglucagon (72-108) Glucagon-like Peptide 1 (GLP-1) Receptor Agonist X
GLPG1205 1445847-37-9 GPR84 Antagonist X X
GLPG3970 2403733-82-2 Compound 88 SIK2/3 Inhibitor X
GLPG4399 SIK3 Inhibitor X
Glyburide Sulfonylurea; Antihyperglycemic Agent X
GM-CSF 83869-56-1 CSF2; Leukine; Sargramostim Cytokine; Immune Modulator X
Go 6983 133053-19-7 PKC (c+n) Inhibitor X
Golimumab Simponi TNFα Inhibitor X
GRP Gastrin-releasing Peptide Stimulates Gastrin Release; Neuropeptide X
GS-441524 1191237-69-0 Metabolite of Remdesivir X
GSK Compound 18 1221277-91-3 LPM029_300303_01 LXR Agonist X
GSK2795039 1415925-18-6 NOX2 Inhibitor X
GSK2801 GSK 2801; KB-146016 BAZ2 Bromodomain Inhibitor X
GSK3326595 1616392-22-3 EPZ015938 PRMT5 Inhibitor X
GSK343 1346704-33-3 EZH2 inhibitor X New – 2025
GSK461364A 929095-18-1 GSK 461364A PLK1 Inhibitor X X
GSK690693 937174-76-0 GSK 690693 AKT Inhibitor X
GSKJ4 1373423-53-0 GSK J4; GTPL8979 Histone Demethylase Inhibitor X X
GW2580 870483-87-7 cFMS Kinase Inhibitor X
GW3965 405911-09-3 LXRα Agonist X
GW501516 317318-70-0 GW-501516 PPARδ Agonist X X X
H-1152 451462-58-1 H1152 ROCK2 Inhibitor X X
H-151 941987-60-6 Antagonist of STING X X New – 2025
H-89 127243-85-0 5-Isoquinolinesulfonamide; Protein Kinase Inhibitor H-89 PKA Inhibitor X
Halobetasol Propionate 66852-54-8 Ulobetasol Glucocorticoid Receptor (GR) Agonist X
hCG Human Chorionic Gonadotropin Luteinizing Hormone; Choriogonadotropin Receptor Agonist X
Hemicholinium Bromide 312-45-8 Hemicholine Choline Transporter (ChT) Inhibitor X
Hesperadin 422513-13-1 Aurora Kinase Inhibitor X
HG-9-91-01 1456858-58-4 Sik Inhibitor 1 SIK1/2/3 Inhibitor X
HGF Hepatocyte Growth Factor c-Met Inhibitor X
Histamine 51-45-6 Histamine Receptor Agonist X
Histamine Phosphate 51-74-1 Histamine Receptor Agonist X
HKLM Heat Killed Listeria monocytogenes TLR2 Agonist X X
Homatropine Bromide 51-56-9 Muscarinic Acetylcholine Receptor (mAChR) Inhibitor X
Human anti-CD73 IgG1 MEDI9447 Anti-CD73 Monoclonal Antibody X
Human IgG1 IgG1 Control Antibody X
Human IgG1 Kappa Immunoglobulin X
Human IgG1 mAb R347 Isotype Control IgG1 Control Antibody X
Human γ-Globulin Serum Fraction X
Hydrochlorothiazide 58-93-5 Diuretic Agent X
Hydrocortisone 50-23-7 17-Hydroxycorticosterone Glucocorticoid Receptor (GR) Agonist X
Hydroxychloroquine Sulfate 747-36-4 Ercoquin; Oxychlorochin; Oxychloroquine; Plaquenil; Toremonil Antimicrobial Agent X
Hydroxyfasudil 155558-32-0 HA 1100 ROCK1, ROCK2 Inhibitor X
Hydroxyurea 127-07-1 Droxia; Hydrea; Hydroxycarbamide; Litalir Antineoplastic Agent; Ribonucleotide Reductase Inhibitor X
Hydroxyzine Dihydrochloride 68-88-2 Arcanax; Neurolax Antihistamine Agent X
Hygromycin B 31282-04-9 Antibiotic Agent X
Iberdomide 1323403-33-3 CC-220 Cereblon (CRBN) E3 ligase modulator X New – 2025
I-BET 1260907-17-2 BET Inhibitor X X
I-BET-151 1300031-49-5 GDK1210151A BET Inhibitor X X X X X
Ibrutinib 936563-96-1 Imbruvica; PCI-32765 BTK Inhibitor X X X X
Ibudilast 50847-11-5 AV-411; Eyevinal; Ibudilastum; Ketas PDE4 Inhibitor X
Ibuprofen 15687-27-1 NeoProfen COX Inhibitor X X
IC-87114 371242-69-2 IC87114 PI3Kδ Inhibitor X X
ICI 63197 27277-00-5 PDE4 Inhibitor X
Idebenone 58186-27-9 Catena; Raxone; Sovrima Synthetic Coenzyme Q10 (CoQ10) Analog X
Idelalisib 870281-82-6 CAL-101; GS-1101; Zydelig PI3Kδ Inhibitor X X X X
IDO-IN-2 914471-09-3 IDO Inhibitor X X X
IFNα 2a IFN-α 2a; INF-α 2a; Interferon α 2a Cytokine X
IFNα 2b IFN-α 2b; INF-α 2b; Interferon α 2b Cytokine X
IFNβ-1b 145155-23-3 Betaseron; INF-β 1b; INFβ 1b; Interferonβ-1b; Interferonβ1b Cytokine X
IFNγ 82115-62-6 Actimmune; Interferon gamma-1b Cytokine X X
IgG4 Isotype IgG4 Control Antibody X X
IKK 16 1186195-62-9 IKK Inhibitor VII; IKK-16 IKK2 Inhibitor X
IKK-2 Inhibitor IV 507475-17-4 IKK2 Inhibitor X
IL-10 130068-27-8 Interleukin 10 Cytokine X X
IL-12 632331-09-0 Interleukin 12 Cytokine X
IL-13 148157-34-0 Interleukin 13 Cytokine X
IL-17A Interleukin 17A Cytokine X X
IL-17F Interleukin 17F Cytokine X
IL-1R Antagonist 566914-00-9 Interleukin 1 Receptor Antagonist IL-1 Receptor Inhibitor X
IL-1β 97599-21-8 Interleukin-1β Cytokine X
IL-2 Aldesleukin; Interleukin 2; Proleukin Cytokine X X
IL-27 Interleukin 27 Cytokine X
IL-29 Interferon λ1; Interleukin 29 Cytokine X
IL-32 Interleukin 32 Cytokine X
IL-33 Interleukin 33 Cytokine X
IL-35 Interleukin 35 Cytokine X
IL-4 207137-56-2 Interleukin 4 Cytokine X
IL-6 Rα CD126 ; Cluster of Differentiation 126 Immunomodulating Agent X
IL-8 CXCL8; Interleukin 8 CXCR1/2 Agonist X
Iloperidone 133454-47-4 Fanapt Antipsychotic Agent X
Iloprost 78919-13-8 Ventavis EP1 Agonist; Prostanoid IP Receptor Agonist X
Imatinib 152459-95-5 Gleevec; Imatinib Methansulfonate; Imatinibum BCR-ABL Inhibitor X X
Indomethacin 53-86-1 Aconip; Indocin; Indometacina; Indometacine; Indometacinum COX Inhibitor X
Infliximab 170277-31-3 Remicade TNFα Inhibitor X X X
Iniparib 160003-66-7 BSI 201 PARP Inhibitor X X
Insulin Aspart Novolog Insulin Receptor Agonist X
Insulin Glargine Lantus Insulin Receptor Agonist X
Insulin Lispro Humalog; Insulin Lispro Recombinant Insulin Receptor Agonist X
IOX1 5852-78-8 Histone Demethylase JMJD Inhibitor X
Ipatasertib 1001264-89-6 GDC-0068, RG7440 ATP-competitive pan-Akt inhibitor X New – 2025
Ipilimumab 477202-00-9 MDX-010; MDX-101; MDX-CTLA-4; MOAB-CTLA-4; Yervoy CTLA-4 Inhibitor X X X
IRAK-1/4 Inhibitor I 509093-47-4 IRAK-1/4 Inhibitor X
Irinotecan 100286-90-6 CPT-11; Campto; Camptosar; Camptothecin-11 DNA Topoisomerase (TOPO) I Inhibitor X X
Irsogladine 57381-26-7 PDE4 Inhibitor X
Isoetharine Mesylate 530-08-5 Isoetarine Mesilate β2 Adrenergic Receptor Agonist X
Isoniazid 54-85-3 Isonicotinic acid hydrazide; Isonicotinsaeurehydrazid; Isonicotinylhydrazine Antibiotic Agent X
Isotretinoin 4759-48-2 13-cis-retinoic acid; Accutane RAR/RXR Agonist X
Istradefylline 155270-99-8 KW-6002 Adenosine A2A Receptor Antagonist X
Itraconazole 84625-61-6 Sporanox Cytochrome P450 51 Inhibitor, Ergosterol Synthesis InhibitorX X X
Ivacaftor 873054-44-5 Kalydeco; VX770 CFTR Potentiator X X
Ivermectin 70288-86-7 MK-933; CD-5024; K-237 inhibitor of Impα/β1-mediated nuclear import; Antiviral towards HIV and the Dengue virus X New – 2025
Ixekizumab Taltz IL-17A Inhibitor X
JAK Inhibitor 1 457081-03-7 CMP 6; Merck-5; Pyridone 6 JAK1 Inhibitor X
JNJ 10191584 Maleate 869497-75-6 VUF6002; Compound 40 Histamine H4 Receptor Antagonist X
JNJ-10397049 708275-58-5 JNJ 10397049 Orexin Receptor Type 2 (OX2) Inhibitor X
JNJ-64619178 2086772-26-9 Onametostat PRMT5 Inhibitor X
JNK Inhibitor VIII 894804-07-0 JNK Inhibitor X
JQ1 1268524-70-4 BET Inhibitor X X X
JWH-015 CB1/2 Agonist X
K252a Multikinase Inhibitor X
KD025 SLx-2119 ROCK2 Inhibitor X
Ketoconazole 65277-42-1 Fungares; Ketoderm; Nizoral; Orifungal M; Panfungol Cytochrome P450 51 Inhibitor X
Ketoprofen 22071-15-4 Actron COX Inhibitor X
Ketotifen Fumarate 34580-14-8 Ketotifen; Ketotifeno; Ketotifenum; Zaditor Antihistamine Agent X
Ki16425 355025-24-0 Ki 16425 LPA1, LPA3 Receptor Inhibitor X
Kisspeptin-10 Metastatin KISS1 Agonist; GPR54 Agonist X
KN93 139298-40-1 CAMKII Inhibitor X X
KNK437 218924-25-5 Hsp Modulator; Hsp Inhibitor (Hsp 72, 73, 90, 105, 27, 40) X
L-744832 1177806-11-9 Farnesyltransferase Inhibitor X
Lansoprazole 103577-45-3 A-65006; AG-1749; Prevacid Proton Pump Inhibitor X
Lapatinib 388082-77-7 GW 572016; Lapatinib Ditosylate; Lapatinib Tosilate Hydrate; Tykerb Tyrosine Kinase Inhibitor (ERBB1, ERBB2) X
L-Arginine Hydrochloride 1119-34-2 Vasodilator X
Larotrectinib 1223403-58-4 Vitrakvi Tropomyosin Kinase Receptor (Trk) Inhibitor X
Leflunomide 75706-12-6 Arava; Leflunomida; Leflunomidum; Lefunomide Dihydroorotate Dehydrogenase (DHODH) Inhibitor X X
Lenalidomide 191732-72-6 Revlimid Immunomodulating Agent; Antineoplastic Agent X X
Lenvatinib 417716-92-8 Lenvima Tyrosine Kinase Inhibitor X X
Letrozole 112809-51-5 CGS 20267; Femara Cytochrome P450 19A1 Inhibitor X
Levamisole Hydrochloride 14769-73-4 (-)-Tetramisole Hydrochloride; Ergamisol; Levamisole HCl; Tramisol Antihelminthic Agent X
LFM-A13 62004-35-7 BTK Inhibitor X
Linezolid 165800-03-3 PNU 100766; Zyvox Antibiotic Agent X
Linsitinib 867160-71-2 OSI-906 IGF-1R Inhibitor X
Liothyronine Liothyronin; Tresitope; Triiodothyronine Thyroid Hormone Receptor Agonist X
Liraglutide Liraglutida; Liraglutidum; Saxenda; Victoza Glucagon-like Peptide 1 (GLP-1) Receptor Agonist X
Lithium Chloride 7447-41-8 Inorganic Compound X X X X
Lofexidine Hydrochloride 21498-08-8 Lucemyra α2A Adrenergic Receptor Agonist X
Lonafarnib 193275-84-2 Sch66336 Ftase Inhbitor X
Lonidamine 50264-69-2 Diclondazolic acid; Doridamina Hexokinase Inhibitor; Glycolysis Inhibitor X
Loperamide Hydrochloride 34552-83-5 Opioid-receptor Agonist X
Lopinavir 192725-17-0 A-157378.0; ABT-378; Aluviran; Koletra Antiretroviral Agent; Protease Inhibitor X
Lorlatinib ALK/ROS1 Inhibitor X
Lornoxicam 70374-39-9 Chlortenoxicam; Xefo NSAID; Analgesic Agent; Anti-inflammatory Agent X
Loteprednol Etabonate 82034-46-6 Alrex; Lotemax Glucocorticoid Receptor (GR) Agonist X
Lovastatin 75330-75-5 Altoprev; Mevacor; Mevinolin HMG-CoA Reductase Inhibitor X
Loxapine Succinate 27833-64-3 Adasuve; Loxitane Antipsychotic Agent X
LP99 Bromodomain Inhibitor X
LPS TLR4 Agonist X X X
Lumacaftor 936727-05-8 VX-809 CFTR Modulator X
Luminespib 747412-49-3 AUY-922; NVP-AUY922 Hsp90 Inhibitor X
lunresertib 2719793-90-3 RP-6306 PKMYT1 Inhibitor X
LY294002 154447-36-6 CK2 Inhibitor; PI3K Inhibitor X X
LY3214996 1951483-29-6 Temuterkib ERK1/ERK2 Inhibitor X
Lysipressin 50-57-7 Lysine vasopressin; [Lys8]-Vasopressin Activates Oxytocin receptors and adenylate-cyclase X New – 2025
M344 251456-60-7 D237; Histone Deacetylase Inhibitor III; MS 344 HDAC Inhibitor X
M5N36 2832887-40-6 Cdc25C inhibitor X New – 2025
Macitentan 441798-33-0 Opsumit ET-A Inhibitor; ET-B Inhibitor X
Manidipine 89226-50-6 Manyper Calcium Channel Blocker; Antihypertensive Agent X
Mavacamten 1642288-47-8 MYK461; SAR439152 Cardiac Myosin activator X
MCC950 NLRP3 Inhibitor X
MCC950 sodium 256373-96-3 CP-456773 sodium; CRID3 sodium salt NLRP3 Inhibitor X
MDV3100 915087-33-1 Enzalutamide; MDV-3100; Xtandi Androgen Receptor (AR) Inhibitor X
Meclocycline Sulfosalicylate 73816-42-9 Meclan; Meclan Cream; Mecloderm; Meclutin Antibiotic Agent X
Medetomidine Hydrochloride 86347-15-1 Domitor; MPV 785; Medetomidine α2 Adrenergic Receptor Agonist X
Medrysone 2668-66-8 HMS; Hydroxymesterone Glucocorticoid Receptor (GR) Agonist X
Mefenamic Acid 61-68-7 CI-473; Ponstel COX Inhibitor X
Megestrol Acetate 595-33-5 Megace; Megestrol; Ovarid Progesterone Receptor (PR) Agonist X
Menadione 58-27-5 Vitamin K3 Phosphatase Inhibitor; Mitochondrial DNA Polymerase γ (pol γ) Inhibitor X
Mepivacaine Hydrochloride 1722-62-9 Carbocaina; Meaverin; Mepivastesin Sodium Channel α Subunit Blocker; Topical Anesthetic Agent X
Mequinol 150-76-5 4-Methoxyphenol; MEHQ Depigmentation Agent X
Mesoridazine Besylate 5588-33-0 Benzenesulfonate; Mesoridazine Antipsychotic Agent X
Metaproterenol Sulfate 5874-97-5 Alupent; Metaprel; Orciprenaline β2 Adrenergic Receptor Agonist X
Metformin Hydrochloride 657-24-9 Haurymellin; Metformina; Metformine Pamoate; Metforminum AMPK Activator; Antihyperglycemic Agent X
Methacholine Chloride Acetyl-beta-methylcholine Chloride; Amechol; Mecholyl Chloride; Methacholine; Provocholine Muscarinic Acetylcholine Receptor Agonist X
Methacycline 3963-95-9 AN100226, BG00002 Inhibitor of epithelial-to-mesenchymal transition EMT X New – 2025
Methapyrilene Hydrochloride 135-23-9 Capathyn; Histadyl; Methacon; Methapyrilene; Methoxylene Antihistamine Agent X
Methazolamide 554-57-4 Naptazane; Neptazane; Neptazaneat Carbonic Anhydrase Inhibitor X
Methocarbamol 532-03-6 Delaxin; Forbaxin; Miolaxin; Neuraxin; Robaxin Muscle Relaxer X
Methotrexate 59-05-2 Abitrexate; Amethopterin; Emtexate; Ledertrexate; MTX; Metoject; Otrexup; Rasuvo Dihydrofolate Reductase (DHFR) Inhibitor X X X
Methyclothiazide 135-07-9 Diuretic; Antihypertensive Agent X
Methyldopa 555-30-6 Aldomet; Alphamethyldopa; Dopamet; Medomet α2 Adrenergic Receptor Agonist X
Methylene Blue 61-73-4 NOS Inhibitor; Guanylate Cyclase Inhibitor X
Mevastatin 73573-88-3 Compactin HMG-CoA Reductase Inhibitor X
Mianserine Hydrochloride 21535-47-7 Bolvidon; Lerivon; Tolvon H1 Receptor Inhibitor; Antidepressant X
Mifamurtide 83461-56-7 Mepact; Mifamurtide Hydrate NOD2 Activator X
Milrinone 78415-72-2 PDE3 Inhibitor X
Mitapivat 1260075-17-9 AG-348 Pyruvate kinase allosteric activator X New – 2025
Mitoglitazone 146062-49-9 CAY10415 Insulin Sensitizer X X
Mitoxantrone Novantrone TOPO II Inhibitor; Antineoplastic Agent X
Mizolastine 108612-45-9 Mizollen H1 Receptor Inhibitor X
Mizoribine 50924-49-7 Bredinin Immunosuppressive Agent; DNA Synthesis Inhibitor X
MK-2206 1032350-13-2 AKT Inhibitor X
MK-8353 1184173-73-6 SCH900353 ERK1/ERK2 Inhibitor X
MK-8457 SYK Inhibitor X
MLN8054 869363-13-3 Aurora Kinase Inhibitor X X
Momelotinib CYT-387; GS-0387 JAK1/2 Inhibitor X X
Mometasone Furoate 83919-23-7 Asmanex; Elomet; Nasonex Glucocorticoid Receptor (GR) Agonist X
Monensin Sodium 22373-78-0 Coban; Rumensin Na+ Ionophore X
Monobenzone 103-16-2 Benoquin; MBEH Skin Whitening Agent X
Monomethyl Fumarate 2756-87-8 GPR109A Agonist X
Montelukast 158966-92-8 MK 0476; MK-0476; Singulair CysLT1 Receptor Inhibitor; GPCR Ligand X
Mosapride Citrate 112885-42-4 AS-4370; DSSTox_CID_26207; Gasmotin 5-HT4 Receptor Agonist X
Motilin Motilin Receptor Agonist X
Moxifloxacin Hydrochloride 186826-86-8 Avalox; Avelox; Moxeza; Vigamox Antimicrobial Agent X
MRL-SYKi DRX_MRL-SYKi SYK Inhibitor X
MRT67307 1190378-57-4 IKKε, MARK1-4, NUAK1 , TBK-1 Inhibitor X X
Mycophenolic Acid 24280-93-1 Cellcept; Melbex; Mycophenolate; Mycophenolsaeure; Myfortic IMPDH Inhibitor X
Myxothiazol 76706-55-3 Cytochrome c Reductase Inhibitor; Mitochondrial Inhibitor X
MZ1 1797406-69-9 BRD4 PROTAC X
N-Acetyl Cysteine 616-91-1 616-91-1; Acetadote; Acetylcysteine; Fluimucil; N-Acetylcysteine Antioxidant X X
Nafcillin Sodium Monohydrate 985-16-0 6-(2-Ethoxy-1-naphthamido)penicillin Antibiotic Agent X
Nalmefene Hydrochloride 58895-64-0 Nalmetrene Opioid Receptor Inhibitor X
Naproxen 22204-53-1 Anaprox; Naprelan; Naprolag; Naprosyn COX Inhibitor X
Natalizumab 189261-10-7 Binds to α4β1-integrin and blocks its interaction X New – 2025
Natalizumab 189261-10-7 AN100226, BG00002 Antibody binds to α4β1-integrin that blocks its interaction with vascular cell adhesion molecule-1 (VCAM-1) X New – 2025
Navitoclax 923564-51-6 ABT-263 Bcl-2 Inhibitor X X
Navoximod 1402836-58-1 GDC-0919; NLG-919; NLG919; RG6078 IDO Inhibitor X X X
Nebivolol 152520-56-4 Bystolic; Lobivon; Nebilet; Nebivololum; R 67555 β1 Adrenergic Receptor Inhibitor X
Nefazodone 83366-66-9 Nefazodona; Nefazodone Hydrochloride; Nefazodonum Antidepressant Agent; 5-HT2A Inhibitor X
Neflamapomid 209410-46-8 VX 745; VX745 p38 MAPK Inhibitor X X
Nefopam Hydrochloride 23327-57-3 Acupan; Ajan; Nefadol; Silentan Non-opioid Analgesic Drug X
Nelarabine 121032-29-9 Arranon DNA Inhibitor X
Neomycin Sulfate 1405-10-3 Fradiomycin; Framycetin; Mycifradin; Soframycin Antibiotic Agent X
Neostigmine Bromide 114-80-7 Eustigmin Bromide; Neo-Proserin; Neoserine Bromide; Proserine Bromide; Prostigmin Acetylcholinesterase Inhibitor X
Nerandomilast 1423719-30-5 BI 1015550 PDE4B Inhibitor X X
Neuromedin B Beta-Neurokinin; Neuromedin K; Porcine Neurokinin B NMBR Agonist X
NI-57 GTPL8573 Bromodomain Inhibitor X
Nialamide 51-12-7 Niamid; Niamide; Nuredal; Surgex Monoamine Oxidase Inhibitor (MAOI) X
Nifuroxazide 965-52-6 RC-27109; SJ000287313 STAT Inhibitor X
Nigericin sodium salt 28643-80-3 Antibiotic Agent / NLRP3 Activator X
Nintedanib 656247-17-5 BIBF 1120; Ofev; Vargatef VEGFR, FGFR, PDGFR Kinase Inhibitor X X
Nirogacestat 1290543-63-3 PF-3084014 γ-secretase inhibitor  X
Nithiamide 140-40-9 Acinitrazole; Aminitrozole Antimicrobial Agent X
Nitrofural 59-87-0 Furacilin; Furacin; Nitrofurazone Antibiotic Agent X
Nitroprusside 13755-38-9 Nipride; Nitroferricyanide; Nitropress Vasodilator X
Nitroxoline 4008-48-4 8-Hydroxy-5-nitroquinoline Antimicrobial agent; Anticancer agent X New – 2025
Nivolumab 946414-94-4 Opdivo PD-1 Inhibitor X X X
Nodinitib-1 799264-47-4 CID-1088438; ML130 NOD1 Inhibitor X
Norethindrone 68-22-4 Norethisterone; Utovlan Progesterone Receptor (PR) Agonist X
Nortriptyline Hydrochloride 72-69-5 Ateben; Avantyl; Demethylamitriptyline; Noritren; Psychostyl; Sensaval SNRI X
Nutlin-3 MDM2 Antagonist X X
NVP-TAE684 761439-42-3 NVP-TAE 684; TAE684 ALK Inhibitor; Kinase Modulator X
NVS1-PAK1-1 DRX_NVS1-PAK1-1 PAK1 Inhibitor X
Obeticholic Acid FXR Agonist X
Octadecanoic acid 57-11-4 Organic Compound X
Odanacatib 603139-19-1 MK0822 Cathepsin K Inhibitor X X
Odevixibat 501692-44-0 A4250 Inhibitor of the ileal bile acid transporter (IBAT) X New – 2025
ODN2006 TLR9 Agonist X X
ODN2395 TLR9 Agonist X
OEA Oleoylethanolamine PPARα Agonist X
Ofloxacin 82419-36-1 Floxin; Ocuflox; Ofloxacine; Tarivid Antimicrobial Agent X
Olaparib 763113-22-0 AZD 2281; AZD-2281; Lynparza PARP Inhibitor X X X
Olcegepant 204697-65-4 BIBN-4096; BIBN 4096BS antagonist of the calcitonin gene-related peptide 1 receptor X New – 2025
Oligomycin A 579-13-5 MCH 32 F0/F1 ATPase Inhibitor; Mitochondrial Inhibitor X X
Olmutinib 1353550-13-6 BI-1482694 Tyrosine Kinase Inhibitor X X X
Omaveloxolone 1474034-05-3 RTA 408 STING Inhibitor X
Omecamtiv Mecarbil 873697-71-3 CK-1827452 Cardiac Myosin activator X
Omeprazole 73590-58-6 Antra; H-168/68; Prilosec Proton Pump Inhibitor X
Omipalisib 1086062-66-9 GSK-2126458; GSK2126458 PI3K Inhibitor; mTOR Inhibitor X X X X
ONC201 DRD2 Inhibitor X X
Oncostatin M 106956-32-5 LIFR-α; OSMR Agonist X
Ondansetron Hydrochloride 99614-02-5 Zofran Antinausea Agent X
ONX 0914 960374-59-8 PR-957 Immunoproteasome Inhibitor X
Orforglipron 2212020-52-3 LY3502970, GLP-1 agonist GLP-1 agonist X New – 2025
Orforglipron 2212020-52-3 LY3502970; GLP-1 receptor agonist 1 GLP-1 agonist X New – 2025
ORIC-944 2369769-29-7 Rinzimetostat Allosteric inhibitor targeting the EED subunit of PRC2 X New – 2025
Orlistat 96829-58-2 Alli; Xenical PI3K Inhibitor; mTOR Inhibitor X
Osimertinib 1421373-65-0 AZD9291; Mereletinib EGFR Inhibitor X X X
OTX015 202590-98-5 MK-8628 BET Inhibitor X X X X
Oxaliplatin 61825-94-3 Diaminocyclohexane Oxalatoplatinum; Eloxatin; L-OHP Antineoplastic Agent; DNA Synthesis Inhibitor X X
Oxaprozin 21256-18-8 Alvo; Daypro; Deflam; Oxaprozine COX Inhibitor X
Oxethazaine 126-27-2 Betalgil; Mucaine; Oxaethacainum; Oxetacaine Local Anaesthetic X
Oxibendazole 20559-55-1 Polymerase Inhibitor X
Oxybuprocaine Hydrochloride 5987-82-6 Benoxinate Hydrochloride Sodium Channel α Subunit Blocker; Topical Anesthetic Agent X
Oxybutynin Chloride 1508-65-2 Ditropan; Oxibutinina; Oxibutyninum; Oxybutynin; Oxytrol Muscarinic Acetylcholine Receptor (mAChR) Inhibitor X
Ozagrel Hydrochloride 78712-43-3 Sodium Ozagrel; UNII-L256JB984D Antiplatelet Agent; Thromboxane A2 Synthesis (TXAS) Inhibitor X
Ozanimod 1306760-87-1 RPC-1063 S1P Receptor Agonist X
P22077 DUB Inhibitor USP47 Inhibitor X
P7C3 301353-96-8 AK340958 NAMPT Activator; Proneurogenic; Neuroprotective X
Paclitaxel 33069-62-4 Anzatax; Asotax; Bristaxol; Praxel; Taxol; Taxol Konzentrat Microtubule Disruptor X X X
Palbociclib 827022-33-3 Ibrance; PD0332991 CDK4/6 Inhibitor X X X
Paliperidone 144598-75-4 Invega Dopamine (D2) Receptor Inhibitor; 5-HT2A Receptor Inhibitor X
Palonosetron Hydrochloride 135729-62-3 Aloxi 5-HT3A Receptor Inhibitor X
Pam3CSK4 TLR1/TLR2 Agonist X
Pamoic Acid Disodium 6640-22-8 Embonic Acid GPR35 Agonist X
Pamrevlumab 946415-13-0 FG-3019 Anti-CTGF
Panitumumab ABX-EGF; Vectibix EGFR Inhibitor X X XZ
Panobinostat 404950-80-7 Faridak; Farydak; LBH-589; LBH589 HDAC Inhibitor X
Paromomycin Sulfate 1263-89-4 Aminosidine Sulfate; Humatin; Paromomycin; Paromomycin Sulfate Salt Antibiotic Agent X
Paroxetine Hydrochloride 110429-35-1 Aropax 20; Paroxat; Paroxetine Hcl SSRI X
Pazopanib 444731-52-6 GW 78603; GW786034; Pazopanibum; Votrient Multi Tyrosine Kinase Receptor Inhibitor (c-KIT, FGFR, PDGFR, VEGFR) X X
PBI-4050 Antifibrotic Agent X X
PD098059 167869-21-8 MEK Inhibitor X
PD123319 130663-39-7 Angiotensin II (AT2) Receptor Inhibitor X
PD184352 212631-79-3 CI-1040 MEK Inhibitor X X
PDGF-BB PDGFRβ Activator X
Pembrolizumab Keytruda PD-1 Inhibitor X X X
Pemetrexed Disodium 150399-23-8 Dihydrofolate Reductase (DHFR) Inhibitor; GAR Transformylase Inhibitor; Thymidylate Synthase Inhibitor X X X
Pemigatinib 1513857-77-6 INCB054828 FGFR Inhibitor X X X
Penciclovir 39809-25-1 Denavir Guanosine Analogue; Antiviral Agent X
Pentamidine 50357-45-4 Nebupent; Pentam Antimicrobial Agent X
Perfluorodecanoic acid 335-76-2 PFDA Reduces mRNA expression of the genes X New – 2025
Pergolide Mesylate 66104-23-2 Pergolide; Pergolide Methanesulfonate; Permax Dopamine Receptor Agonist X
Perindopril Erbumine 107133-36-8 Aceon Angiotensin-converting Enzyme Inhibitor X
Pertuzumab 2C4 Antibody; MOAB 2C4; Omnitarg; Perjeta; rhuMAb-2C4 HER2 Dimerization Inhibitor X
PF-04217903 956905-27-4 c-Met Inhibitor X
PF-06297470 mGluR5 Inhibitor X
PF-06650833 1817626-54-2 IRAK4 Inhibitor X
PFI-1 1403764-72-6 PF-06405761; PF-6405761 BET Inhibitor X X X
PFI-3 SMARCA2/4 Inhibitor; Polybromo 1 (PBRM1) Inhibitor X X
PFI-4 PFI4 Bromodomain Inhibitor X
PHA-408 503555-55-3 IKK2 Inhibitor X
Phenazopyridine Hydrochloride 136-40-3 Bisteril; Mallophene; Phenazopyridine HCl; Urodine Sodium Channel α Subunit Blocker; Topical Anesthetic Agent X
Pheniramine Maleate 132-20-7 Avil-retard; Daneral; Inhiston; Naphcon; Trimetose Antihistamine Agent X
Phenylbutazone 50-33-9 Butatron; Butazolidin COX Inhibitor X
Phenylephrine Cyclomydril; Mydfrin α1 Adrenergic Receptor Agonist X
Phorbol 12-myristate 13-acetate 16561-29-8 PMA PKC Activator X
Piclamilast 144035-83-6 Cpodpmb; RP 73401 PDE4 Inhibitor X
Picropodophyllin 477-47-4 AXL1717; Picropodophyllotoxin Microtubule Disruptor X
PIM447 1210608-43-7 LGH447 PIM Kinase Inhibitor X
Pimasertib 1236699-92-5 AS 703026; AS703026 MEK Inhibitor X
Pimobendan 74150-27-9 Vetmedin PDE3 Inhibitor X
Pioglitazone 111025-46-8 Actos; Glustin; Pioglitazona; Pioglitazonum PPARγ Agonist X
Pirfenidone 53179-13-8 Esbriet; Etuary; KitosCell; Pirespa; Pirfenex Antifibrotic Agent X X
Pironetin 151519-02-7 Microtubule Disruptor X
Pirtobrutinib 2101700-15-4 LOXO-305 BTK Inhibitor X
Pitolisant 362665-56-3 Tiprolisant Histamine H3 Receptor Inverse Agonist X
Pizotifen Malate Pizotyline; Sandomigran 5-HT Receptor Antagonist X
PKN1/2-IN-1 942425-34-5 Cell penetrant and selective PKN2 (PRK2) inhibitor X X New – 2025
Pladienolide B 445493-23-2 Spliceosome Inhibitor X X X
Plerixafor 155148-31-5 AMD 3100 CXCR4 Inhibitor X X X
PLX4720 918505-84-7 PLX-4720 BRAF Inhibitor X
PNU 74654 113906-27-7 Wnt/β-catenin Pathway Inhibitor X
Poly(I:C)HMW TLR3 Agonist X X
Pomalidomide 19171-19-8 3-amino Thalidomide; CC-4047 Immunomodulating Agent; Antineoplastic Agent X
Ponatinib 3-amino Thalidomide; AP 24534; AP24534; Iclusig BCR-ABL Inhibitor X X
Posaconazole 171228-49-2 Noxafil; Sch 56592 CYP51 Inhibitor X
PP1 172889-26-8 Mutant Kinases Inhibitor II; PP1 Analog II Src Family Inhibitor X
PP242 1092351-67-1 PP 242 mTOR Inhibitor X
Pralatrexate 146464-95-1 Folotyn DHFR Inhibitor X
Pralsetinib 2097132-94-8 BLU-667 RET Inhibitor X X X
Pramlintide 151126-32-8 High affinity for amylin, CGRP and calcitonin receptors X New – 2025
Pramoxine Hydrochloride 637-58-1 Topical Anesthetic X
Pranlukast 103177-37-3 Onon Cysteinyl Leukotriene Receptor 1 (CYSLTR1) Antagonist X
Praziquantel 55268-74-1 Biltricide Antimicrobial Agent X
Prednisolone 50-24-8 Hydroretrocortine; Metacortandralone; Millipred; Omnipred; Orapred; PRDL; Pediapred; Prednisolona Glucocorticoid Receptor (GR) Agonist X X
Prednisone 53-03-2 Adasone; Dehydrocortisone; Deltasone; Meticorten; Prednisonum Glucocorticoid Receptor (GR) Agonist X
Pregnenolone sulfate sodium salt 1852-38-6 3β-Hydroxy-5-pregnen-20-one monosulfate sodium Inhibitor of cannabinoid CB1 receptor X New – 2025
Prilocaine Hydrochloride 721-50-6 Citanest Anaesthetic Agent X
Primaquine Diphosphate 90-34-6 NSC 149765; Tronolane Quinone Reductase 2 Inhibitor X
Probenecid 57-66-9 Benecid; Benemid; Probalan; Probecid; Probenecid Acid Uricosuric Agent X X
Procarbazine Hydrochloride 671-16-9 Matulane; Nathulane; Natunalar; PROCARBAZINE HCl Antineoplastic Agent X
Progesterone 57-83-0 Prometrium Progesterone Receptor (PR) Agonist X
Prostaglandin D2 41598-07-6 PGD2 DP Agonist X
Prostaglandin E2 363-24-6 Cervidil; Dinoprostone; Prepidil; Prostin E2 EP Agonist X
PrRP-31 Prolactin Releasing Peptide-31 hGR3/GPR10 Agonist X
PRT062607 PRT-062607 Syk Inhibitor X
Psilocybin 2641522-10-1 Tryptamine, hallucinogenic X X X X New – 2025
Pyridostigmine Bromide 101-26-8 Kalimin; Mestinon; Mestinon Bromide; Regonol Cholinesterase Inhibitor X
Pyrithioxin 1098-97-1 1098-97-1; Bonifen; Encefabol; Pyrithioxine; Pyritinol Neurotropic Agent X
QRFP-26 P518 GPR 103 Agonist X
Quinacrine Dihydrochloride Dihydrate 83-89-6 Atabrine Hydrochloride PLA2 (phophoslipase A2) Inhibitor X
Quizartinib 950769-58-1 AC220 FLT3 Inhibitor X
R(-)rolipram 85416-73-5 Adeo; Rolipramum; ZK 62711 PDE4 Inhibitor X
RA11740397 (MLI2) LRRK2 Inhibitor X
Radicicol 12772-57-5 Monorden HSP90 Inhibitor X X
Raltitrexed 112887-68-0 Tomudex; ZD1694 Dihydrofolate Reductase Inhibitor; Thymidylate Synthase Inhibitor X
Rapamycin 53123-88-9 AY 22989; Rapamune; SILA 9268A; Sirolimus; WY-090217 mTOR Inhibitor X X X X
RDEA119 923032-37-5 BAY 869766; RDEA-119; Refametinib MEK Inhibitor X
Reboxetine Mesylate 98769-84-7 Noradrenalin Uptake Inhibitor X
Regorafenib 755037-03-7 BAY 73-4506 Multikinase Inhibitor (VEGFR2-TIE2 Tyrosine Kinase) X
Remdesivir 1809249-37-3 GS-5734 Nucleoside Analogue X
Repaglinide 135062-02-1 GlucoNorm; NovoNorm; Prandin; Repaglinidum Antidiabetic Agent X
Resatorvid 243984-11-4 TAK-242, CLI-095 Toll-like receptor 4 (TLR4) inhibitor X New – 2025
Resiquimod 144875-48-9 TLR7/TLR8 Agonist X
Resmetirom 920509-32-6 MGL-3196, VIA-3196 TRH Receptor B-Agonist X X New – 2025
Resveratrol 501-36-0 CYP1A1 Inhibitor X X
Retapamulin 224452-66-8 Altabax; Altargo Antimicrobial Agent X
Retinol 68-26-8 Vitamin A X
rhM-CSF Not Listed Recombinant Human Macrophage-colony Stimulating Factor M-CSF Receptor Agonist X
Ribociclib 1211441-98-3 LEE01 CDK4/6 Inhibitor X
Rimonabant 158681-13-1 SR141716 CB1 Inverse Agonist; GPCR Ligand X
Riociguat 625115-55-1 Adempas sGC Activator X
Risdiplam 1825352-65-5 RG7916; RO7034067 SMN2 pre-mRNA splicing modifier X New – 2025
Risedronate Sodium 115436-72-1 Actonel; Atelvia; Benet Biphosphonate; Bone Density Conservation Agent X
Ritlecitinib 1792180-81-4 PF-06651600 JAK3 inhibitor X New – 2025
Ritonavir 155213-67-5 A-84538; ABT-53; ABT-538; Abbott 84538; Norvir HIV Protease Inhibitor X
RN486 1242156-23-5 BTK Inhibitor X
Ro 106-9920 62645-28-7 Ubiquitin Ligase Inhibitor X
Ro 20-1724 29925-17-5 PDE4 Inhibitor X
Ro 320-1195 Not Listed p38 MAPK Inhibitor X
Ro 32-0432 151342-35-7 PKC (c+n) Inhibitor X
Ro 5126766 946128-88-7 RO5126766 BRAF Inhibitor; MEK Inhibitor X
Rofecoxib 162011-90-7 Ceoxx; MK 966; Vioxx COX-2 Inhibitor X X
Roflumilast 162401-32-3 Daliresp; Daxas; ROF; Roflumilastum PDE4 Inhibitor X X
Roflumilast N-Oxide 292135-78-5 PDE4 Inhibitor X X
Rolipram 61413-54-5 Adeo; Rolipramum; ZK 62711 PDE4 Inhibitor X
Romidepsin 128517-07-7 FK 228 HDAC Inhibitor X
Rosiglitazone 122320-73-4 TZD; Avandia PPARγ Agonist X X X
Rosuvastatin 287714-41-4 Rosuvastatin; Crestor HMG-CoA Reductase Inhibitor X
Rotenone 83-79-4 Barbasco; Dactinol; Paraderil; Tubatoxin Mitochondrial Inhibitor; NADH Dehydrogenase Inhibitor X
Roxadustat Not Listed FG-4592 HIF-PHI Inhibitor X
Rucaparib Phosphate 459868-92-9 PARP Inhibitor X
Ruxolitinib 941678-49-5 INCB018424; Jakafi JAK1/2 Inhibitor X X X X
RVU120 1609452-30-3 SEL120; SEL120-34A CDK8 Inhibitor X X
RXDX-106 Not Listed TAM Receptor Inhibitor X
R-α-Methylhistamine 6986-90-9 H3 Histamine Receptor Agonist X
S31-201 501919-59-1 Nsc 74859 STAT3 Inhibitor X
Salbutamol Sulfate 51022-70-9 Albuterol β2 Adrenergic Receptor Agonist X
Salicylanilide 87-17-2 2-Hydroxybenzanilide; N-Phenylsalicylamide Antimicrobial Agent X
Salicylic Acid 69-72-7 2-Carboxyphenol; 2-Hydroxybenzoic acid; O-hydroxybenzoic acid COX Inhibitor X
Salinomycin Monosodium 55721-31-8 Coxistac; Salinomycin P-glycoprotein 1 Inhibitor X
Salmeterol Xinafoate 94749-08-3 Arial; Asmerole; Salmetedur; Serevent Diskus β2 Adrenergic Receptor Agonist X X
Saracatinib 379231-04-6 AZD 0530; AZD0530 Src/Abl Inhibitor X X
Sarafloxacin Hydrochloride 91296-87-6 Antimicrobial Agent X
Saxagliptin 361442-04-8 Onglyza DPP-4 Inhibitor; Antidiabetic Agent X
SB203580 152121-47-6 p38 MAPK Inhibitor X
SB431542 301836-41-9 TGFβR1 Kinase Inhibitor; ALK Inhibitor X X X X
SB525334 Not Listed TGFβ RI Kinase Inhibitor VIII TGFβR1 Kinase Inhibitor; ALK Inhibitor X
SB939 929016-96-6 Pracinostat HDAC Inhibitor X
SC-514 354812-17-2 IKK2 Inhibitor X
Scriptaid 287383-59-9 Scriptide HDAC Inhibitor X
Secukinumab 1229022-83-6 Cosentyx IL-17A Inhibitor X
Selinexor 1393477-72-9 KPT-330 CRM1 Inhibitor X
Selnoflast 2260969-36-4 Somalix; RO-7486967; IZD334 NLRP3 Inhibitor X
Selonsertib 1448428-04-3 ASK1 Inhibitor X X
Selumetinib 606143-52-6 ARRY-142886; AZD6244 MEK Inhibitor X X
Semagacestat 425386-60-3 LY450139 γ-Secretase Inhibitor X
Semaglutide 910463-68-2 GLP-1 Analogue X
Serotonin Not Listed 5-HT; 5-Hydroxytryptamine; Antemovis; Enteramine Monoamine Neurotransmitter X
Sertraline 79617-96-2 Zoloft SSRI X
SGC-CBP30 Not Listed CREBBP/EP300 Bromodomain Inhibitor X X
SGC-I-CBP112 Not Listed CBP/p300 Bromodomain Inhibitor X
SGI-1776 1025065-69-3 Pim Kinase Inhibitor IX PIM Kinase Inhibitor X
Shaoguamycin B 2738-64-9 Piericidin A; Piericidin A1; Piericidine A Mitochondrial Inhibitor; NADH Dehydrogenase Inhibitor X
Shikonin 517-89-5 C.I. 75535; Isoarnebin 4 inhibitor of TMEM16A chloride channel, pyruvate kinase M2, TNF-α, and NF-κB pathway X New – 2025
Sildenafil Citrate 171599-83-0 Viagra PDE5 Inhibitor X X
Simvastatin 79902-63-9 Zocor HMG-CoA Reductase Inhibitor X X
Sirolimus 53123-88-9 Rapamycin; AY-22989; NSC 226080 mTOR inhibitor X New – 2025
SL 327 305350-87-2 MEK Inhibitor X
SLPI Not Listed Antileukoproteinase; ALK1; ALP; BLPI; HUSI; HUSI-I; MPI; WAP4; WFDC4 Peptidase Inhibitor Protein X
SNS-314 1057249-41-8 Aurora Kinase Inhibitor X
Sodium Hydroxide 1310-73-2 Caustic Soda; Lye; Sodium Hydrate Inorganic Compound X
Somatostatin 28 Not Listed Cyclic tetradecapeptide Somatostatin Receptor Agonist X
Sonidegib 956697-53-3 Smoothened (SMO) Inhibitor X
Sorafenib Tosylate 475207-59-1 BAY 43-9006; Nexavar; Tosylate Salt Multikinase Inhibitor (RAF/VEGFR-2/PDGFRβ) X X X
Sotagliflozin 1018899-04-1 Zynquista; LX4211 SGLT1/SGLT2 Inhibitor X
SP600125 129-56-6 1,9-Pyrazoloanthrone JNK Inhibitor X
Sparsentan 254740-64-2 RE-021; DARA-a Angiotensin II and endothelin A receptor antagonist X New – 2025
SPD-304 Not Listed TNFα Inhibitor X
Sphingosine-1-phosphate 26993-30-6 C18-Sphingosine 1-phosphate; D-erythro-Sphingosine-1-phosphate S1P Receptor Agonist X
Spiramycin 8025-81-8 Rovamycine Antimicrobial Agent X
Spironolactone 52-01-7 52-01-7; Aldactone; Spiroctan; Spirolactone; Verospiron Aldosterone Inhibitor X
SR2211 Not Listed RORγ Inhibitor X
SR31747 132173-07-0 Sigma Ligand X
SRT2104 Not Listed “for BioSeek” Sirtuin Modulator SIRT1 Activator X
ssRNA40 Not Listed R-1075 TLR8 Agonist X X
STA 5326 541550-19-0 Apilimod IL-12/IL-23 Inhibitor X
Staurosporine 62996-74-1 AM-2282; STS Multikinase Inhibitor X X X
SU6656 330161-87-0 Src Family Inhibitor X
Succinate Not Listed Succinic Acid Chemical Intermediate X
Sulfasalazine 599-79-1 Azopyrin; Colo-Pleon; Salazosulfapyridine; Salicylazosulfapyridine; Sulcolon Anti-inflammatory Agent X
Sulforaphane Not Listed Phytochemical; Antioxidant; Detoxifying Enzyme Inducer X
Sunitinib Malate 341031-54-7 SU011248; SU11248; Sutent Multikinase Inhibitor (VEGFR2, CSF-1R, PDGFR, SCFR, FLT3, RET) X X X
Suzetrigine 2649467-58-1 VX-548 NaV1.8 inhibitor that acts as an analgesic, blocker of sodium channel protein X New – 2025
SX-682 1648843-04-2 Allosteric inhibitor of CXCR1 and CXCR2 X New – 2025
Synta66 Not Listed CLC001531 CRAC Channel Inhibitor X
T0901317 293754-55-9 T 0901317 LXR Agonist; FXR Agonist X X
Tacrolimus 104987-11-3 FK-506; FR900506; NCGC00179232-01 Calcineurin Inhibitor; FK506-binding Protein 1A Inhibitor X X
Tadalafil 171596-29-5 ADCIRCA; Cialis; Ic351; Tadanafil PDE5 Inhibitor X
Tafamidis 594839-88-0 TTR Stabilizer X
Tafenoquine 106635-81-8 Krintafel Antimalarial Agent X
Talazoparib 1207456-01-6 Talzenna PARP Inhibitor X X
Tamoxifen 10540-29-1 Genox; Nolvadex; Soltamox; Tamifen Estrogen Receptor Modulator X
Tanespimycin 75747-14-7 17-AAG Hsp90 Inhibitor X X
Tapinarof 79338-84-4 WBI-1001; Benvitimod; GSK2894512 AhR Agonist X X
Taurolithocholic Acid 6042-32-6 G Protein-coupled Bile Acid Receptor 1 Agonist X
Tavapadon 1643489-24-0 PF-06649751; CVL-751 Agonist of dopamine D1/D5 receptor X New – 2025
Tazemetostat 1403254-99-8 EPZ-6438 EZH2 inhibitor X New – 2025
Teicoplanin 61036-62-2 Targocid; Ticosin Antibiotic Agent X
Telaglenastat 1439399-58-2 CB-839 GLS1 Inhibitor X X
Telbivudine 3424-98-4 Epavudine; Sebivo; Tyzeka Antiviral Agent; Thymidine β-L-nucleoside Analogue X
Telmisartan 144701-48-4 BIBR 277; Micardis Angiotensin II (AT2) Receptor Inhibitor X X
Temsirolimus 162635-04-3 CCI 779; Torisel FK506-binding Protein 1A (FKBP1A) Inhibitor; mTOR Inhibitor X
Tenidap 120210-48-2 9K7CJ74ONH; Tenidapum 5-Lipoxygenase Inhibitor; COX1/2 Inhibitor X
Tepotinib 1100598-32-0 EMD-1214063 c-Met Inhibitor X
Terbinafine 91161-71-6 Lamasil; Lamisil; Lamisil AT; SF-86-327; Terbinex Antimicrobial Agent X
Teriflunomide 108605-62-5 A771726; Aubagio; Flucyamide; HMR1726 Pyrimidine Synthesis Inhibitor; DHODH Inhibitor X
Tetracycline Hydrochloride 60-54-8 Abramycin; Achromycin; Deschlorobiomycin; Tetracyclinum; Tsiklomitsin Antibiotic Agent X
TGFβ Not Listed TGFβRI/II Agonist X
TGFβ2 Not Listed TGFRI, TGFRII Agonist X
TGFβ3 Not Listed TGFRI, TGFRII Agonist X
TGF-βRI Kinase Inhibitor 396129-53-6 TGFβR1 Kinase Inhibitor X
TGX-221 663619-89-4 Tgx 221 PI3Kβ Inhibitor X
Thapsigargin 67526-95-8 SERCA Inhibitor X X
Thiostrepton 1393-48-2 Alaninamide; Antibiotic A 8506; Antibiotic X 146; Bryamycin; Thiactin Oligopeptide Antibiotic X
Tianeptine Sodium 30123-17-2 Coaxil; Stablon; Tatinol Tricyclic Antidepressant X
Tigecycline 220620-09-7 GAR-936; TBG-MINO; Tygacil; WAY-GAR-936 Antibiotic Agent X
Tilorone Dihydrochloride 27591-69-1 Antiviral Agent; Type I Interferon Inducer X X X
Tin Protoporphyrin IX 14325-05-4 NSC 267099 Heme Oxygenase Inhibitor X
Tin(II) Chloride 7772-99-8 Stannous Chloride; Tin Protochloride; Tin Salt Chemical Compound X
Tioxolone 4991-65-5 Thioxolone Carbonic Anhydrase Inhibitor X
Tipiracil HCl 183204-72-0 Thymidine Phosphorylase Inhibitor X
Tiratricol 51-24-1 Triac Thyroid Hormone Analogue; Physiologic Thyroid Hormone X
Tivozanib 475108-18-0 AV-951; KRN951 VEGFR Inhibitor X
TMP-153 128831-46-9 Acetyl-coA Cholesterol Acyltransferase (ACAT) Inhibitor X
TNP-470 129298-91-5 AGM-1470; Agm 1470; DRG-0148 Antineoplastic Agent X
Tofacitinib 477600-75-2 Tasocitinib; Tofacitinibum; Xeljanz JAK1/3 Inhibitor X X X X
Topotecan Hydrochloride 119413-54-6 Hycamptamine; Hycamtin; SKF S-104864-A TOPO I Inhibitor X X
Torcetrapib 262352-17-0 CP 529414; CP-529414 CETP Inhibitor X
Torin-1 1222998-36-8 Torin1 mTOR Inhibitor X X
Torin-2 1223001-51-1 Torin2 mTOR Inhibitor X X
Torsemide 56211-40-6 Demadex; TORSEMIDE; Torasemida; Torasemidum Diuretic Agent X
Tozadenant 870070-55-6 SYN-115 Adenosine A2a Receptor Inhibitor X X X
Trametinib 871700-17-3 GSK1120212; Mekinist MEK Inhibitor X X X
Tranexamic Acid 1197-18-8 Cyklokapron; Tranexamsaeure Plasminogen Inhibitor X
Tranilast 53902-12-8 Rizaben Antiallergic Agent X X
Trans-Triprolidine 486-12-4 Antihistamine Agent X
Trastuzumab 180288-69-1 Herceptin; Herclon HER2/neu Receptor Inhibitor X
Trastuzumab deruxtecan 1826843-81-5 DS-8201; DS-8201a Anti-HER2 Drug Conjugate X
Treprostinil 81846-19-7 UT-15 DP1/EP2 Agonist X X
Tretinoin 302-79-4 ATRA; Aberela; Retinoic Acid; Trans-Retinoic Acid; Vitamin A Acid; all-trans-Retinoic Acid RAR/RXR Agonist X
Triamcinolone 124-94-7 Glucocorticoid Receptor (GR) Agonist X
Tribanibulin 897016-82-9 Klisyri Tubulin Inhibitor X X
Trichostatin A 58880-19-6 58880-19-6; TSA; Trichostatin HDAC Inhibitor X
Triflusal 322-79-2 Aflex; Disgren; Grendis; Triflux Platelet Antiaggregant X
Trigonelline 535-83-1 Trigenolline Nrf2 inhibitor X New – 2025
Trilostane 13647-35-3 13647-35-3; Desopan; Trilostano; Trilostanum; Vetoryl 3 β-Hydroxysteroid Dehydrogenase Inhibitor X
Tropine 120-29-6 3-Tropanol Atropine Precursor X
Trypan Blue 72-57-1 Direct Blue 14; Membraneblue; TRYPAN BLUE; UNII-I2ZWO3LS3; VisionBlue Diazo Dye X
Tubastatin A 1252003-15-8 HDAC Inhibitor X
Tucatinib 937263-43-9 Irbinitinib, ARRY-380, ONT-380 Selective HER2 inhibitor X New – 2025
Tunicamycin 11089-65-9 Antibiotic Agent X
TWEAK Human TWEAK; TNF-like Weak Inducer; TNFSF12 Cytokine X
Tyr[SO3H]27)-CCK8 25126-32-3 C-Terminal Octapeptide of Cholecystokinin (CCK); Kinevac; Sincalide Stimulates Pancreatic Secretion X
Tyrphostin AG 1296 146535-11-7 AG-1296 PDGFR Inhibitor X
U-75302 119477-85-9 Leukotriene B4 (LTB4) Receptor Inhibitor X
UK 14, 304 Not Listed α2 Adrenergic Receptor Agonist X
Umbralisib 1532533-67-7 TGR-1202; RP5264 PI3Kδ/CK1ε Inhibitor X
Umifenovir 131707-25-0 Antiviral X X
UNC0642 Not Listed G9a and GLP Inhibitor X
UNC2025 1429881-91-3 Mer Inhibitor; FLT3 Inhibitor X
UO126 109511-58-2 U0126 MEK Inhibitor X
Upadacitinib 1310726-60-3 ABT-494 JAK1 Inhibitor X X
Urolithin A Not Listed Microflora Metabolite X
Ursodeoxycholic Acid 128-13-2 Actigall; Delursan; Ursodiol; Ursolvan Bile Acid X
Ursolic Acid 77-52-1 Urson; Malol; Prunol Cosmetic Additive X
Ustekinumab 815610-63-0 Anti-Human IL-12/IL-23, Human Antibody anti-IL-12/IL-23 IgG1κ human monoclonal antibody
UTP Not Listed Uridine triphosphate Nucleotide  X
Vadimezan 117570-53-3 5,6-Mexaa; DMXAA DT-Diaphorase Inhibitor X X
Valdecoxib 181695-72-7 Bextra COX2 Inhibitor X
Valinomycin 2001-95-8 Antibiotic Agent X
Valnemulin Hydrochloride 133868-46-9 Pleuromutilin Antibiotic X
Valproic Acid 1069-66-5 Depakene; Depakine; Dipropylacetic acid HDAC Inhibitor; GABA Transaminase Inhibitor X X
Vamorolone 13209-41-1 VBP15 dissociative steroidal anti-inflammatory agent and membrane-stabilizer X
Vandetanib 443913-73-3 AZD6474; Caprelsa; ZD6474 VEGFR2, EGFR Inhibitor X X
Vardenafil 330808-88-3 Levitra; Staxyn; Vardenafilum PDE5 Inhibitor X
Vasopressin Not Listed ADH; AVP; Antidiuretic Hormone; Argipressin Vasopressin Receptor Agonist X
Vegetable Extract HI_V19 Not Listed Vegetable Extract X
VEGF-165 127464-60-2 VEGF Receptor Agonist X
Vemurafenib 1029872-54-5 BRAF(V600E) Kinase Inhibitor; PLX4032; RO5185426; Zelboraf BRAF Inhibitor X X
Venetoclax 1257044-40-8 ABT199; GDC-0199; Venclexta Bcl-2 Inhibitor X X X X X
Vepdegestrant 2229711-68-4 ARV-471 PROTAC estrogen receptor degrader= X New – 2025
Verapamil 52-53-9 CP-165331; Calan; Covera-hs; Iproveratril; Isoptin; Tarka; Verelan L-type Calcium Channel Blocker X
Vinblastine 865-21-4 VLB; Vincaleukoblastine Microtubule Disruptor X
Vincristine Sulfate 2068-78-2 Leurocristine; Vincristin; Vincristina; Vincristine; Vincristinum Microtubule Disruptor X
Vinorelbine 71486-22-1 Exelbine; Navelbine; UNII-Q6C979R91Y; Vinorelbina; Vinorelbinum Microtubule Inhibitor X
Vinpocetine 42971-09-5 Apovincaminic Acid Ethyl Ester; Cavinton; TCV-3B PDE1 Inhibitor X
Vismodegib 879085-55-9 Erivedge; GDC-0449 Hedgehog Pathway Inhibitor X X X
Vitamin D2 50-14-6 Vitamin D Receptor (VDR) Agonist X
VLX1570 1431280-51-1 DUB Inhibitor X
Vorasidenib 1644545-52-7 AG-881 mIDH1/2 inhibitor X New – 2025
Vorinostat 149647-78-9 SAHA; Suberoylanilide Hydroxamic Acid; Zolinza HDAC Inhibitor (HDAC1, HDAC2, HDAC3, HDAC6) X X
Voxtalisib 1123889-87-1 PI3K-IN-1; XL765 PI3K Inhibitor; mTOR Inhibitor X
VX702 479543-46-9 VX 702 p38 MAPK Inhibitor X
VZ185 2306193-61-1 BRD7/9 PROTAC Degrader X
WKYMVm-NH2 Not Listed BDBM86297 Formyl Peptide Receptor (FPR1, FPR2) Agonist X
Wortmannin 19545-26-7 Antibiotic SL-2052; KY 12420; SL-2052; Wartmannin PI3Kinase Inhibitor X
WS6 1421227-53-3 EBP1/IKK Inhibitor X
XAV939 284028-89-3 Tankyrase (TNKS) Inhibitor X X X X
XL019 945755-56-6 JAK2 Inhibitor X
XL147 956958-53-5 PI3K Inhibitor X; Pilaralisib PI3K Inhibitor X
XL880 849217-64-7 EXEL-2880; Foretinib; GSK089; GSK1363089; XL-880 VEGFR2 Inhibitor X X X X
Y27632 146986-50-7 ROCK1, ROCK2 Inhibitor X X
YM155 781661-94-7 Survivin Inhibitor X
YM201636 371942-69-7 PIKfyve Inhibitor X
Zaprinast 37762-06-4 PDE5/PDE6/PDE9 Inhibitor X
Zegocractin 1713240-67-5 CM-4620 CRAC Inhibitor X X
Zetomipzomib 1629677-75-3 KZR-616 Immunoproteasome Inhibitor X
Zinc Chloride 7646-85-7 Chemical Compound X
Zinc Protoporphyrin IX 15442-64-5 ZPP Heme Oxygenase Inhibitor X
Ziprasidone Hydrochloride 122883-93-6 Zeldox; Ziprasidone Antipsychotic Agent X
Ziritaxestat 1628260-79-6 GLPG1690 Autotaxin Inhibitor X X
ZM39923 273727-89-2 JAK3 Inhibitor X
ZM449829 4452-06-6 JAK3 Inhibitor X
Zoldonrasib 2922732-54-3 RMC-9805 2nd generation K-Ras Inhibitor X New – 2025
Zongertinib 2728667-27-2 BI 1810631 HER2 and EGFR tyrosine kinase inhibitor X New – 2025
Zunsemetinib 1640282-42-3 ATI-450; CDD-450 MK2 Inhibitor X
α-Amanitin 23109-05-9 Alpha-Amanitine; Alpha-Amatoxin; HSDB 3458 RNA Polymerase II Inhibitor X
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