Biological Information
No. of Assays on Panel:
132
Assays on Panel:
Family
GPCR
Name
NK1 Human Tachykinin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
100
Protein
NK1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
5-HT2C Human Serotonin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
1003
Protein
5-HT2C
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
5-HT4E Human Serotonin GPCR Cell Based Agonist cAMP LeadHunter Assay - FR
Item
1044
Protein
5-HT4
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
5-HT4E Human Serotonin GPCR Cell Based Antagonist cAMP LeadHunter Assay - FR
Item
1045
Protein
5-HT4
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
Y1 Human Neuropeptide Y GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
106
Protein
Y1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
NT1 Human Neurotensin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
109
Protein
NT1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
M3 Human Acetylcholine (Muscarinic) GPCR Cell Based Agonist Calcium Flux LeadHunter Assay - FR
Item
1243
Protein
M3
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
M3 Human Acetylcholine (Muscarinic) GPCR Cell Based Antagonist Calcium Flux LeadHunter Assay - FR
Item
1244
Protein
M3
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
M1 Human Acetylcholine (Muscarinic) GPCR Cell Based Agonist Calcium Flux LeadHunter Assay - FR
Item
1262
Protein
M1
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
GAL2 Human Galanin GPCR Cell Based Agonist Calcium Flux LeadHunter Assay - FR
Item
1292
Protein
GAL2
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
alpha2A Human Adrenoceptor GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
13
Protein
alpha2A
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
5-HT1A Human Serotonin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
131
Protein
5-HT1A
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
D2S Human Dopamine GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
1322
Protein
D2
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
5-HT2B Human Serotonin GPCR [125I](±)DOI Binding Agonist Radioligand LeadHunter Assay - FR
Item
1333
Protein
5-HT2B
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
5-HT2C Human Serotonin GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
137
Protein
5-HT2C
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
D2L Human Dopamine GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
1405
Protein
D2
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
5-HT6 Human Serotonin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
142
Protein
5-HT6
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
5-HT7 Human Serotonin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
144
Protein
5-HT7
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
M1 Human Acetylcholine (Muscarinic) GPCR Cell Based Antagonist Calcium Flux LeadHunter Assay - FR
Item
1474
Protein
M1
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
alpha1A Human Adrenoceptor GPCR Cell Based Agonist Calcium Flux LeadHunter Assay - FR
Item
1500
Protein
alpha1A
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
alpha1A Human Adrenoceptor GPCR Cell Based Antagonist Calcium Flux LeadHunter Assay - FR
Item
1501
Protein
alpha1A
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
MT1 Human Melatonin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
1538
Protein
MT1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
5-HT2B Human Serotonin GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
1609
Protein
5-HT2B
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
NT1 Human Neurotensin GPCR Cell Based Agonist Calcium Flux LeadHunter Assay - FR
Item
1612
Protein
NT1
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
5-HT6 Human Serotonin GPCR Cell Based Agonist cAMP LeadHunter Assay - FR
Item
1627
Protein
5-HT6
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
5-HT6 Human Serotonin GPCR Cell Based Antagonist cAMP LeadHunter Assay - FR
Item
1628
Protein
5-HT6
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
NT1 Human Neurotensin GPCR Cell Based Antagonist Calcium Flux LeadHunter Assay - FR
Item
1634
Protein
NT1
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
M2 Human Acetylcholine (Muscarinic) GPCR Cell Based Agonist cAMP LeadHunter Assay - FR
Item
1658
Protein
M2
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
M2 Human Acetylcholine (Muscarinic) GPCR Cell Based Antagonist cAMP LeadHunter Assay - FR
Item
1659
Protein
M2
Organism
Human
Assay Sub Type
Cell Based
Family
Ion Channel
Name
KV (Non-Selective) Rat Potassium Ion Channel [125I] alpha-Dendrotoxin Binding LeadHunter Assay - FR
Item
166
Protein
Kv1.1
Organism
Rat
Assay Sub Type
Binding
Family
GPCR
Name
5-HT7 Human Serotonin GPCR Cell Based Agonist cAMP LeadHunter Assay - FR
Item
1661
Protein
5-HT7
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
5-HT7 Human Serotonin GPCR Cell Based Antagonist cAMP LeadHunter Assay - FR
Item
1662
Protein
5-HT7
Organism
Human
Assay Sub Type
Cell Based
Family
Ion Channel
Name
SKCa (Non-Selective) Rat Potassium Ion Channel [125I] Apamin Binding LeadHunter Assay - FR
Item
167
Protein
SKCa
Organism
Rat
Assay Sub Type
Binding
Family
GPCR
Name
M4 Human Acetylcholine (Muscarinic) GPCR Cell Based Agonist cAMP LeadHunter Assay - FR
Item
1670
Protein
M4
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
M4 Human Acetylcholine (Muscarinic) GPCR Cell Based Antagonist cAMP LeadHunter Assay - FR
Item
1671
Protein
M4
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
D1 Human Dopamine GPCR Cell Based Agonist cAMP LeadHunter Assay - FR
Item
1685
Protein
D1
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
D1 Human Dopamine GPCR Cell Based Antagonist cAMP LeadHunter Assay - FR
Item
1686
Protein
D1
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
MT2 Human Melatonin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
1687
Protein
MT2
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
D5 Human Dopamine GPCR Cell Based Agonist cAMP LeadHunter Assay - FR
Item
1688
Protein
D5
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
D5 Human Dopamine GPCR Cell Based Antagonist cAMP LeadHunter Assay - FR
Item
1689
Protein
D5
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
GAL2 Human Galanin GPCR Cell Based Antagonist Calcium Flux LeadHunter Assay - FR
Item
1893
Protein
GAL2
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
AT1 Human Angiotensin GPCR Cell Based Agonist Calcium Flux LeadHunter Assay - FR
Item
1912
Protein
AT1
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
AT1 Human Angiotensin GPCR Cell Based Antagonist Calcium Flux LeadHunter Assay - FR
Item
1913
Protein
AT1
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
sst1 Human Somatostatin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
1940
Protein
sst1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
CT Human Calcitonin GPCR Cell Based Agonist cAMP LeadHunter Assay - FR
Item
1964
Protein
CT
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
CT Human Calcitonin GPCR Cell Based Antagonist cAMP LeadHunter Assay - FR
Item
1965
Protein
CT
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
beta2 Human Adrenoceptor GPCR Cell Based Agonist cAMP LeadHunter Assay - FR
Item
1976
Protein
beta2
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
beta2 Human Adrenoceptor GPCR Cell Based Antagonist cAMP LeadHunter Assay - FR
Item
1977
Protein
beta2
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
A1 Human Adenosine GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
2
Protein
A1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
beta2 Human Adrenoceptor GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
20
Protein
beta2
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
sst5 Human Somatostatin GPCR Cell Based Agonist cAMP LeadHunter Assay - FR
Item
2087
Protein
sst5
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
sst5 Human Somatostatin GPCR Cell Based Antagonist cAMP LeadHunter Assay - FR
Item
2088
Protein
sst5
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
MT2 Human Melatonin GPCR Cell Based Agonist cAMP LeadHunter Assay - FR
Item
2092
Protein
MT2
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
sst4 Human Somatostatin GPCR Cell Based Agonist cAMP LeadHunter Assay - FR
Item
2095
Protein
sst4
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
MT2 Human Melatonin GPCR Cell Based Antagonist cAMP LeadHunter Assay - FR
Item
2100
Protein
MT2
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
sst4 Human Somatostatin GPCR Cell Based Antagonist cAMP LeadHunter Assay - FR
Item
2103
Protein
sst4
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
beta3 Human Adrenoceptor GPCR Cell Based Agonist cAMP LeadHunter Assay - FR
Item
2189
Protein
beta3
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
NK1 Human Tachykinin GPCR Cell Based Agonist Calcium Flux LeadHunter Assay - FR
Item
2190
Protein
NK1
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
beta3 Human Adrenoceptor GPCR Cell Based Antagonist cAMP LeadHunter Assay - FR
Item
2191
Protein
beta3
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
NK1 Human Tachykinin GPCR Cell Based Antagonist Calcium Flux LeadHunter Assay - FR
Item
2192
Protein
NK1
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
sst1 Human Somatostatin GPCR Cell Based Agonist cAMP LeadHunter Assay - FR
Item
2253
Protein
sst1
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
sst1 Human Somatostatin GPCR Cell Based Antagonist cAMP LeadHunter Assay - FR
Item
2254
Protein
sst1
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
alpha1A Human Adrenoceptor GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
2338
Protein
alpha1A
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
AT1 Human Angiotensin GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
24
Protein
AT1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
AT2 Human Angiotensin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
26
Protein
AT2
Organism
Human
Assay Sub Type
Binding
Family
Lipid Metabolism
Name
PLA2 (Group V, Non-Selective) Human Phospholipase A2 Enzymatic LeadHunter Assay - FR
Item
3176
Protein
Organism
Human
Assay Sub Type
Enzymatic
Family
GPCR
Name
5-HT2A Human Serotonin GPCR Cell Based Agonist IP1 LeadHunter Assay - FR
Item
3196
Protein
5-HT2A
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
5-HT2C Human Serotonin GPCR Cell Based Agonist IP1 LeadHunter Assay - FR
Item
3197
Protein
5-HT2C
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
5-HT2A Human Serotonin GPCR Cell Based Antagonist IP1 LeadHunter Assay - FR
Item
3198
Protein
5-HT2A
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
5-HT2C Human Serotonin GPCR Cell Based Antagonist IP1 LeadHunter Assay - FR
Item
3199
Protein
5-HT2C
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
5-HT2B Human Serotonin GPCR Cell Based Agonist IP1 LeadHunter Assay - FR
Item
3344
Protein
5-HT2B
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
5-HT2B Human Serotonin GPCR Cell Based Antagonist IP1 LeadHunter Assay - FR
Item
3345
Protein
5-HT2B
Organism
Human
Assay Sub Type
Cell Based
Family
Transmembrane (Other)
Name
sigma2 Human Binding Agonist Radioligand LeadHunter Assay - FR
Item
3468
Protein
Organism
Human
Assay Sub Type
Binding
Family
Enzyme
Name
Monoamine Oxidase B (MAO-B) Human Enzymatic LeadHunter Assay - FR
Item
3477
Protein
MAO-B
Organism
Human
Assay Sub Type
Enzymatic
Family
Enzyme
Name
Acetylcholinesterase Human Enzymatic LeadHunter Assay - FR
Item
363
Protein
AChE
Organism
Human
Assay Sub Type
Enzymatic
Family
GPCR
Name
mGlu5 Human Glutamate (Metabotropic) GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
3844
Protein
mGlu5
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
A2A Human Adenosine GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
4
Protein
A2A
Organism
Human
Assay Sub Type
Binding
Family
PDE
Name
PDE4A1A Human Phosphodiesterase Enzymatic LeadHunter Assay - FR
Item
4074
Protein
PDE4A
Organism
Human
Assay Sub Type
Enzymatic
Family
PDE
Name
PDE4B1 Human Phosphodiesterase Enzymatic LeadHunter Assay - FR
Item
4076
Protein
PDE4B
Organism
Human
Assay Sub Type
Enzymatic
Family
Enzyme
Name
PDE4D2 Human Phosphodiesterase Enzymatic LeadHunter Assay - FR
Item
4077
Protein
PDE4D
Organism
Human
Assay Sub Type
Enzymatic
Family
GPCR
Name
GAL2 Human Galanin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
410
Protein
GAL2
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
5-HT3 Human Serotonin Ion Channel Binding Antagonist Radioligand LeadHunter Assay - FR
Item
411
Protein
5-HT3A
Organism
Human
Assay Sub Type
Binding
Family
Enzyme
Name
COX2 Human Cyclooxygenase Enzymatic LeadHunter Assay - FR
Item
4186
Protein
COX2
Organism
Human
Assay Sub Type
Enzymatic
Family
GPCR
Name
M5 Human Acetylcholine (Muscarinic) GPCR Cell Based Agonist Calcium Flux LeadHunter Assay - FR
Item
4217
Protein
M5
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
M5 Human Acetylcholine (Muscarinic) GPCR Cell Based Antagonist Calcium Flux LeadHunter Assay - FR
Item
4218
Protein
M5
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
GAL1 Human Galanin GPCR Cell Based Agonist Calcium Flux LeadHunter Assay - FR
Item
4257
Protein
GAL1
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
GAL1 Human Galanin GPCR Cell Based Antagonist Calcium Flux LeadHunter Assay - FR
Item
4258
Protein
GAL1
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
sst2 Human Somatostatin GPCR Cell Based Agonist Calcium Flux LeadHunter Assay - FR
Item
4304
Protein
sst2
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
sst2 Human Somatostatin GPCR Cell Based Antagonist Calcium Flux LeadHunter Assay - FR
Item
4305
Protein
sst2
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
sst3 Human Somatostatin GPCR Cell Based Agonist Calcium Flux LeadHunter Assay - FR
Item
4308
Protein
sst3
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
sst3 Human Somatostatin GPCR Cell Based Antagonist Calcium Flux LeadHunter Assay - FR
Item
4309
Protein
sst3
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
A1 Human Adenosine GPCR Cell Based Agonist Calcium Flux LeadHunter Assay - FR
Item
4314
Protein
A1
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
A1 Human Adenosine GPCR Cell Based Antagonist Calcium Flux LeadHunter Assay - FR
Item
4315
Protein
A1
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
alpha2A Human Adrenoceptor GPCR Cell Based Agonist Calcium Flux LeadHunter Assay - FR
Item
4316
Protein
alpha2A
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
alpha2A Human Adrenoceptor GPCR Cell Based Antagonist Calcium Flux LeadHunter Assay - FR
Item
4317
Protein
alpha2A
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
5-HT1A Human Serotonin GPCR Cell Based Agonist Calcium Flux LeadHunter Assay - FR
Item
4332
Protein
5-HT1A
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
5-HT1A Human Serotonin GPCR Cell Based Antagonist Calcium Flux LeadHunter Assay - FR
Item
4333
Protein
5-HT1A
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
5-HT1B Human Serotonin GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
4376
Protein
5-HT1B
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
5-HT1B Human Serotonin GPCR Cell Based Agonist cAMP LeadHunter Assay - FR
Item
4385
Protein
5-HT1B
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
5-HT1B Human Serotonin GPCR Cell Based Antagonist cAMP LeadHunter Assay - FR
Item
4386
Protein
5-HT1B
Organism
Human
Assay Sub Type
Cell Based
Family
Transporter
Name
SERT Human Serotonin Transporter Binding Antagonist Radioligand LeadHunter Assay - FR
Item
439
Protein
SERT
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
D1 Human Dopamine GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
44
Protein
D1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
A1 Human Adenosine GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
442
Protein
A1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
A2B Human Adenosine GPCR Cell Based Agonist cAMP LeadHunter Assay - FR
Item
452
Protein
A2B
Organism
Human
Assay Sub Type
Cell Based
Family
Ion Channel
Name
Cav1.2 (L-type) Human Calcium Ion Channel Binding (Verapamil Site) LeadHunter Assay - FR
Item
4524
Protein
Cav1.2 (L-type)
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
Cav1.2 (L-type) Human Calcium Ion Channel Binding (diltiazem site) (benzothiazepines) LeadHunter Assay - FR
Item
4549
Protein
Cav1.2 (L-type)
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
A2B Human Adenosine GPCR Cell Based Antagonist cAMP LeadHunter Assay - FR
Item
455
Protein
A2B
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
D2S Human Dopamine GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
46
Protein
D2
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
5-HT2A Human Serotonin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
471
Protein
5-HT2A
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
D3 Human Dopamine GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
48
Protein
D3
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
sst4 Human Somatostatin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
482
Protein
sst4
Organism
Human
Assay Sub Type
Binding
Family
Transporter
Name
DAT Human Dopamine Transporter Functional Antagonist Uptake LeadHunter Assay - FR
Item
4865
Protein
DAT
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
D4.4 Human Dopamine GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
49
Protein
D4
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
A2B Human Adenosine GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
5
Protein
A2B
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
D5 Human Dopamine GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
50
Protein
D5
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
5-HT4E Human Serotonin GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
501
Protein
5-HT4
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
KATP Rat Potassium Ion Channel Mass Spectrometry Binding Antagonist Ligand LeadHunter Assay - FR
Item
5111
Protein
Organism
Rat
Assay Sub Type
Binding
Family
Ion Channel
Name
Cav1.2 (L-type) Human Calcium Ion Channel Binding (Dihydropyridine Site) LeadHunter Assay - FR
Item
5538
Protein
CaV1.2 (DHP site)
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
A3 Human Adenosine GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
6
Protein
A3
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
GAL1 Human Galanin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
62
Protein
GAL1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
sst5 Human Somatostatin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
626
Protein
sst5
Organism
Human
Assay Sub Type
Binding
Family
NHR
Name
PPARalpha Human NHR Binding Agonist Radioligand LeadHunter Assay - FR
Item
640
Protein
PPARalpha
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
D3 Human Dopamine GPCR Cell Based Agonist cAMP LeadHunter Assay - FR
Item
683
Protein
D3
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
D3 Human Dopamine GPCR Cell Based Antagonist cAMP LeadHunter Assay - FR
Item
684
Protein
D3
Organism
Human
Assay Sub Type
Cell Based
Family
Transmembrane (Other)
Name
sigma1 Human Binding Agonist Radioligand LeadHunter Assay - FR
Item
889
Protein
sigma1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
M1 Human Acetylcholine (Muscarinic) GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
91
Protein
M1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
M2 Human Acetylcholine (Muscarinic) GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
93
Protein
M2
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
M3 Human Acetylcholine (Muscarinic) GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
95
Protein
M3
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
M4 Human Acetylcholine (Muscarinic) GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
96
Protein
M4
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
M5 Human Acetylcholine (Muscarinic) GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
97
Protein
M5
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
A3 Human Adenosine GPCR Cell Based Agonist cAMP LeadHunter Assay - FR
Item
982
Protein
A3
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
A3 Human Adenosine GPCR Cell Based Antagonist cAMP LeadHunter Assay - FR
Item
983
Protein
A3
Organism
Human
Assay Sub Type
Cell Based
Testing Information
Test Sample Requirements:
Minimum for Screen : 190 µl of 10mM stock -OR- 1 mg (pre-weighed) for 10µM final testing.
Turnaround Time
Standard:
15 Business Days
Additional Information
Brand:
LeadHunter
Testing Location:
France - Celle L'Evescault