Biological Information
No. of Assays on Panel:
44
Assays on Panel:
Family
GPCR
Name
5-HT4E Human Serotonin GPCR Cell Based Agonist cAMP LeadHunter Assay - FR
Item
1044
Protein
5-HT4
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
5-HT4E Human Serotonin GPCR Cell Based Antagonist cAMP LeadHunter Assay - FR
Item
1045
Protein
5-HT4
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
delta (DOP) Human Opioid GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
114
Protein
delta (DOP)
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
5-HT1A Human Serotonin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
131
Protein
5-HT1A
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
D2S Human Dopamine GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
1322
Protein
D2
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
H3 Human Histamine GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
1332
Protein
H3
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
beta1 Human Adrenoceptor GPCR Cell Based Agonist cAMP LeadHunter Assay - FR
Item
1605
Protein
beta1
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
beta1 Human Adrenoceptor GPCR Cell Based Antagonist cAMP LeadHunter Assay - FR
Item
1606
Protein
beta1
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
5-HT6 Human Serotonin GPCR Cell Based Antagonist cAMP LeadHunter Assay - FR
Item
1628
Protein
5-HT6
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
5-HT7 Human Serotonin GPCR Cell Based Antagonist cAMP LeadHunter Assay - FR
Item
1662
Protein
5-HT7
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
D1 Human Dopamine GPCR Cell Based Antagonist cAMP LeadHunter Assay - FR
Item
1686
Protein
D1
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
beta1 Human Adrenoceptor GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
18
Protein
beta1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
H3 Human Histamine GPCR Cell Based Agonist cAMP LeadHunter Assay - FR
Item
1800
Protein
H3
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
H3 Human Histamine GPCR Cell Based Antagonist cAMP LeadHunter Assay - FR
Item
1801
Protein
H3
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
5-HT1D Rat Serotonin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
1974
Protein
5-HT1D
Organism
Rattus norvegicus (Rat)
Assay Sub Type
Binding
Family
GPCR
Name
beta2 Human Adrenoceptor GPCR Cell Based Agonist cAMP LeadHunter Assay - FR
Item
1976
Protein
beta2
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
beta2 Human Adrenoceptor GPCR Cell Based Antagonist cAMP LeadHunter Assay - FR
Item
1977
Protein
beta2
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
A2A Rat Adenosine GPCR Cell Based Antagonist cAMP LeadHunter Assay - FR
Item
2056
Protein
A2A
Organism
Rat
Assay Sub Type
Cell Based
Family
GPCR
Name
beta3 Human Adrenoceptor GPCR Cell Based Agonist cAMP LeadHunter Assay - FR
Item
2189
Protein
beta3
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
beta3 Human Adrenoceptor GPCR Cell Based Antagonist cAMP LeadHunter Assay - FR
Item
2191
Protein
beta3
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
H1 Human Histamine GPCR Cell Based Agonist Calcium Flux LeadHunter Assay - FR
Item
2542
Protein
H1
Organism
Human
Assay Sub Type
Cell Based
Family
Ion Channel
Name
nAChR (alpha7) Human Ion Channel Binding Antagonist Radioligand LeadHunter Assay - FR
Item
3010
Protein
nAChR
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
nAChR (alpha4/beta2) Human Ion Channel Binding Agonist Radioligand LeadHunter Assay - FR
Item
3029
Protein
nAChR
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
GABAA (alpha1/beta2/gamma2) Human Ion Channel [3H] Muscimol Binding Agonist Radioligand LeadHunter Assay - FR
Item
3051
Protein
GABAA
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
5-HT2A Human Serotonin GPCR Cell Based Agonist IP1 LeadHunter Assay - FR
Item
3196
Protein
5-HT2A
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
beta3 Human Adrenoceptor GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
3963
Protein
beta3
Organism
Homo sapiens (Human)
Assay Sub Type
Binding
Family
GPCR
Name
A1 Human Adenosine GPCR Cell Based Agonist Calcium Flux LeadHunter Assay - FR
Item
4314
Protein
A1
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
delta (DOP) Human Opioid GPCR Cell Based Agonist Calcium Flux LeadHunter Assay - FR
Item
4328
Protein
delta (DOP)
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
5-HT1A Human Serotonin GPCR Cell Based Agonist Calcium Flux LeadHunter Assay - FR
Item
4332
Protein
5-HT1A
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
5-HT1A Human Serotonin GPCR Cell Based Antagonist Calcium Flux LeadHunter Assay - FR
Item
4333
Protein
5-HT1A
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
5-HT1B Human Serotonin GPCR Cell Based Agonist cAMP LeadHunter Assay - FR
Item
4385
Protein
5-HT1B
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
A1 Human Adenosine GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
442
Protein
A1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
kappa (KOP) Human Opioid GPCR Cell Based Agonist Calcium Flux LeadHunter Assay - FR
Item
4459
Protein
kappa (KOP)
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
kappa (KOP) Human Opioid GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
4461
Protein
kappa (KOP)
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
GABAA (alpha1/beta2/gamma2) Human Ion Channel [3H] Flunitrazepam Binding Agonist Radioligand LeadHunter Assay - FR
Item
4518
Protein
GABAA(BZD site)
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
Cav1.2 (L-type) Human Calcium Ion Channel Binding (Verapamil Site) LeadHunter Assay - FR
Item
4524
Protein
Cav1.2 (L-type)
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
Cav1.2 (L-type) Human Calcium Ion Channel Binding (diltiazem site) (benzothiazepines) LeadHunter Assay - FR
Item
4549
Protein
Cav1.2 (L-type)
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
5-HT2A Human Serotonin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
471
Protein
5-HT2A
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
5-HT4E Human Serotonin GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
501
Protein
5-HT4
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
KATP Rat Potassium Ion Channel Mass Spectrometry Binding Antagonist Ligand LeadHunter Assay - FR
Item
5111
Protein
Organism
Rat
Assay Sub Type
Binding
Family
Ion Channel
Name
GluK2 Human Ion Channel [3H] Kainic acid Binding LeadHunter Assay - FR
Item
5379
Protein
Kainate
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
Sodium Channel Site2 (Non-selective) Rat Ion Channel Batrachotoxin Mass Spectrometry Binding LeadHunter Assay - FR
Item
5572
Protein
Nav1.5
Organism
Rat
Assay Sub Type
Binding
Family
Ion Channel
Name
Glutamate (NMDA, NR1/NR2A) Human Ion Channel [3H] CGP-39653 Binding LeadHunter Assay - FR
Item
5875
Protein
GluN1 / GluN2A
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
Glutamate (AMPA, Non-Selective) Rat Ion Channel [3H] AMPA Binding LeadHunter Assay - FR
Item
64
Protein
AMPA
Organism
Rat
Assay Sub Type
Binding
Testing Information
Test Sample Requirements:
Minimum for Screen : 120 µl of 10mM stock -OR- 1 mg (pre-weighed) for 10µM final testing.
Turnaround Time
Standard:
15 Business Days
Additional Information
Brand:
LeadHunter
Testing Location:
France - Celle L'Evescault