OVERVIEW
DOCUMENTS/REFERENCES
Biological Information
No. of Assays on Panel:
170
Assays on Panel:
Family
GPCR
Name
A1 Human Adenosine GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
200510
Protein
A1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
A2A Human Adenosine GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
200610
Protein
A2A
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
A2B Human Adenosine GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
200650
Protein
A2B
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
A3 Human Adenosine GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
200720
Protein
A3
Organism
Human
Assay Sub Type
Binding
Family
Transporter
Name
Adenosine Human Transporter Binding Antagonist Radioligand LeadHunter Assay - TW
Item
202020
Protein
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
alpha1A Human Adrenoceptor GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
203110
Protein
alpha1A
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
alpha1B Human Adrenoceptor GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
203210
Protein
alpha1B
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
alpha1D Human Adrenoceptor GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
203400
Protein
alpha1D
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
alpha2A Human Adrenoceptor GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
203630
Protein
alpha2A
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
alpha2B Human Adrenoceptor GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
203710
Protein
alpha2B
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
alpha2C Human Adrenoceptor GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
203810
Protein
alpha2C
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
beta1 Human Adrenoceptor GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
204010
Protein
beta1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
beta2 Human Adrenoceptor GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
204110
Protein
beta2
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
beta3 Human Adrenoceptor GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
204200
Protein
beta3
Organism
Human
Assay Sub Type
Binding
Family
Transporter
Name
NET Human Norepinephrine Transporter Binding Antagonist Radioligand LeadHunter Assay - TW
Item
204410
Protein
NET
Organism
Human
Assay Sub Type
Binding
Family
NHR
Name
AR Human Androgen NHR Binding Agonist Radioligand LeadHunter Assay - TW
Item
206000
Protein
AR
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
AT1 Human Angiotensin GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
210030
Protein
AT1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
AT2 Human Angiotensin GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
210120
Protein
AT2
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
APJ Human Apelin GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
210720
Protein
APJ
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
BB1 Human Bombesin GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
211600
Protein
BB1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
BB2 Human Bombesin GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
211700
Protein
BB2
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
BB3 Human Bombesin GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
211800
Protein
BB3
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
B1 Human Bradykinin GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
212520
Protein
B1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
B2 Human Bradykinin GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
212620
Protein
B2
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
CGRP (CLR/RAMP1) Human Calcitonin GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
214020
Protein
CLR
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
Cav1.2 (L-type) Rat Calcium Ion Channel Binding (Diltiazem Site) LeadHunter Assay - TW
Item
214510
Protein
Cav1.2 (L-type)
Organism
Rat
Assay Sub Type
Binding
Family
Ion Channel
Name
Cav1.2 (L-type) Human Calcium Ion Channel Binding (Dihydropyridine Site) LeadHunter Assay - TW
Item
214610
Protein
Cav1.2 (L-type)
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
Cav1.2 (L-type) Rat Calcium Ion Channel Binding (Verapamil Site) LeadHunter Assay - TW
Item
215000
Protein
Cav1.2 (L-type)
Organism
Rat
Assay Sub Type
Binding
Family
Ion Channel
Name
Cav2.2 (N-type) Rat Calcium Ion Channel Binding Antagonist Radioligand LeadHunter Assay - TW
Item
216000
Protein
Cav2.2 (N-type)
Organism
Rat
Assay Sub Type
Binding
Family
Ion Channel
Name
Cav2.2 (N-type) Human Calcium Ion Channel [3H] Gabapentin Binding Antagonist Radioligand LeadHunter Assay - TW
Item
216020
Protein
Cav2.2 (N-type)
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
CB1 Human Cannabinoid GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
217050
Protein
CB1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
CB2 Human Cannabinoid GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
217100
Protein
CB2
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
CCR1 Human Chemokine GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
217510
Protein
CCR1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
CCR2 Human Chemokine GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
217550
Protein
CCR2
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
CCR5 Rhesus Macaque Chemokine GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
217730
Protein
CCR5
Organism
Rhesus Macaque
Assay Sub Type
Binding
Family
GPCR
Name
CCK1 (CCKA) Human Cholecystokinin GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
218030
Protein
CCK1 (CCKA)
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
CCK2 (CCKB) Human Cholecystokinin GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
218130
Protein
CCK2 (CCKB)
Organism
Human
Assay Sub Type
Binding
Family
Transporter
Name
CHT1 Human Choline Transporter Binding Antagonist Radioligand LeadHunter Assay - TW
Item
219010
Protein
CHT1
Organism
Human
Assay Sub Type
Binding
Family
Cytoskeleton
Name
Tubulin Rat [3H] Colchicine Binding LeadHunter Assay - TW
Item
219100
Protein
Organism
Rat
Assay Sub Type
Binding
Family
GPCR
Name
CRF1 Human Corticotropin-Releasing Factor GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
219150
Protein
CRF1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
D1 Human Dopamine GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
219500
Protein
D1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
D2L Human Dopamine GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
219600
Protein
D2
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
D2S Human Dopamine GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
219700
Protein
D2
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
D3 Human Dopamine GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
219800
Protein
D3
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
D4.4 Human Dopamine GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
220000
Protein
D4
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
D5 Human Dopamine GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
220200
Protein
D5
Organism
Human
Assay Sub Type
Binding
Family
Transporter
Name
DAT Human Dopamine Transporter Binding Antagonist Radioligand LeadHunter Assay - TW
Item
220320
Protein
DAT
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
ETA Human Endothelin GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
224010
Protein
ETA
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
ETB Human Endothelin GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
224110
Protein
ETB
Organism
Human
Assay Sub Type
Binding
Family
Kinase
Name
EGFR Human RTK Kinase Binding Radiometric LeadHunter Assay [10 uM ] - TW
Item
225510
Protein
EGFR
Organism
Human
Assay Sub Type
Binding
Family
NHR
Name
ERalpha Human Estrogen NHR Binding Agonist Radioligand LeadHunter Assay - TW
Item
226010
Protein
ERalpha
Organism
Human
Assay Sub Type
Binding
Family
NHR
Name
ERbeta Human Estrogen NHR Binding Agonist Radioligand LeadHunter Assay - TW
Item
226050
Protein
ERbeta
Organism
Human
Assay Sub Type
Binding
Family
Transporter
Name
GABA (Non-Selective) Rat Transporter Binding Antagonist Radioligand LeadHunter Assay - TW
Item
226400
Protein
Organism
Rat
Assay Sub Type
Binding
Family
Ion Channel
Name
GABAA (Non-Selective) Rat Ion Channel [3H] Muscimol Binding Agonist Radioligand LeadHunter Assay - TW
Item
226500
Protein
Organism
Rat
Assay Sub Type
Binding
Family
Ion Channel
Name
GABAA (Non-Selective) Rat Ion Channel [3H] Flunitrazepam Binding Agonist Radioligand LeadHunter Assay - TW
Item
226600
Protein
Organism
Rat
Assay Sub Type
Binding
Family
Ion Channel
Name
GABAA (Non-Selective) Rat Ion Channel [3H] Ro-15-1788 Binding (Hippocampus) LeadHunter Assay - TW
Item
226630
Protein
Organism
Rat
Assay Sub Type
Binding
Family
Ion Channel
Name
GABAA (Non-Selective) Rat Ion Channel [3H] TBOB Binding Antagonist Radioligand LeadHunter Assay - TW
Item
226810
Protein
Organism
Rat
Assay Sub Type
Binding
Family
GPCR
Name
GABAB (B1a/B2) Human GABAB GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
228610
Protein
GABAB (B1/B2)
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
GABAB (B1b/B2) Human GABAB GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
228710
Protein
GABAB (B1/B2)
Organism
Human
Assay Sub Type
Binding
Family
Cell Surface (Other)
Name
GHB Rat Binding Antagonist Radioligand LeadHunter Assay - TW
Item
231650
Protein
Organism
Rat
Assay Sub Type
Binding
Family
GPCR
Name
Glucagon Human Glucagon GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
231680
Protein
GCGR
Organism
Human
Assay Sub Type
Binding
Family
NHR
Name
GR Human Glucocorticoid NHR Binding Agonist Radioligand LeadHunter Assay - TW
Item
232030
Protein
GR
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
Glutamate (AMPA, Non-Selective) Rat Ion Channel [3H] AMPA Binding LeadHunter Assay - TW
Item
232600
Protein
Organism
Rat
Assay Sub Type
Binding
Family
Ion Channel
Name
Glutamate (Kainate, Non-Selective) Rat Ion Channel [3H] Kainic acid Binding LeadHunter Assay - TW
Item
232710
Protein
Organism
Rat
Assay Sub Type
Binding
Family
Ion Channel
Name
Glutamate (NMDA, NR1/NR2A) Human Ion Channel [3H] CGP-39653 Binding LeadHunter Assay - TW
Item
232820
Protein
GluN1/ GluN2A
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
Glutamate (NMDA, Non-Selective) Rat Ion Channel [3H] MDL 105,519 Binding LeadHunter Assay - TW
Item
232910
Protein
Organism
Rat
Assay Sub Type
Binding
Family
Ion Channel
Name
Glutamate (Non-Selective) Rat Ion Channel [3H] TCP Binding LeadHunter Assay - TW
Item
233000
Protein
Organism
Rat
Assay Sub Type
Binding
Family
Ion Channel
Name
Glutamate (NMDA, Non-Selective) Rat Ion Channel [3H] Ifenprodil Binding LeadHunter Assay - TW
Item
234000
Protein
Organism
Rat
Assay Sub Type
Binding
Family
GPCR
Name
mGlu2 Human Glutamate (Metabotropic) GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
236400
Protein
mGlu2
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
mGlu5 Human Glutamate (Metabotropic) GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
237000
Protein
mGlu5
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
Glycine alpha1 Human Ion Channel [3H] Strychnine Binding LeadHunter Assay - TW
Item
239010
Protein
GLRA1
Organism
Human
Assay Sub Type
Binding
Family
Transporter
Name
GLYT1 Rat Glycine Transporter uptake LeadHunter Assay - TW
Item
239110-1
Protein
GLYT1
Organism
Rat
Assay Sub Type
Cell Based
Family
GPCR
Name
GnRH Human Gonadotrophin-Releasing Hormone GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
239200
Protein
GnRH
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
GHSR Human Ghrelin GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
239300
Protein
GHSR
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
H1 Human Histamine GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
239610
Protein
H1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
H2 Human Histamine GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
239710
Protein
H2
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
H3 Human Histamine GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
239820
Protein
H3
Organism
Human
Assay Sub Type
Binding
Family
Transmembrane (Other)
Name
Imidazoline I2 Central Rat Binding Antagonist Radioligand LeadHunter Assay - TW
Item
241000
Protein
Organism
Rat
Assay Sub Type
Binding
Family
Kinase
Name
IR (INSR) Rat RTK Kinase Binding Radiometric LeadHunter Assay Agonist Radioligand - TW
Item
243000
Protein
IR
Organism
Rat
Assay Sub Type
Binding
Family
Cell Surface (Other)
Name
IL-1 R1 Human Interleukin Binding Agonist Radioligand LeadHunter Assay - TW
Item
243530
Protein
IL-1R-1
Organism
Human
Assay Sub Type
Binding
Family
Cell Surface (Other)
Name
IL-6 Human Interleukin Binding Agonist Radioligand LeadHunter Assay - TW
Item
244100
Protein
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
CXCR1 (IL-8RA) Human Chemokine GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
244420
Protein
CXCR1 (IL-8RA)
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
CXCR2 (IL-8RB) Human Chemokine GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
244500
Protein
CXCR2 (IL-8RB)
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
CXCR4 Human Chemokine GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
244550
Protein
CXCR4
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
CX3CR1 Human Chemokine GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
244600
Protein
CX3CR1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
CysLT1 Human Leukotriene GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
250460
Protein
CysLT1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
MCH1 Human Melanin-Conc. Hormone GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
251010
Protein
MCH1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
MCH2 Human Melanin-Conc. Hormone GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
251050
Protein
MCH2
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
MC1 Human Melanocortin GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
251100
Protein
MC1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
MC3 Human Melanocortin GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
251300
Protein
MC3
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
MC4 Human Melanocortin GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
251350
Protein
MC4
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
MC5 Human Melanocortin GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
251400
Protein
MC5
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
MT1 Human Melatonin GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
251600
Protein
MT1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
MT2 Human Melatonin GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
251700
Protein
MT2
Organism
Human
Assay Sub Type
Binding
Family
Transporter
Name
VMAT (Non-Selective) Human Vesicular Monoamine Transporter Binding LeadHunter Assay - TW
Item
252030
Protein
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
Motilin Human Motilin GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
252200
Protein
Motilin
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
M1 Human Acetylcholine (Muscarinic) GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
252610
Protein
M1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
M2 Human Acetylcholine (Muscarinic) GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
252710
Protein
M2
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
M3 Human Acetylcholine (Muscarinic) GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
252810
Protein
M3
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
M4 Human Acetylcholine (Muscarinic) GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
252910
Protein
M4
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
M5 Human Acetylcholine (Muscarinic) GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
253010
Protein
M5
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
Acetylcholine (Muscarinic, Non-Selective) Rat GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
254000
Protein
Organism
Rat
Assay Sub Type
Binding
Family
GPCR
Name
NK1 Human Tachykinin GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
255520
Protein
NK1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
NK2 Human Tachykinin GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
255620
Protein
NK2
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
NK3 Human Tachykinin GPCR Binding (Agonist Radioligand) Assay, Panlabs
Item
255710
Protein
NK3
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
Y1 Human Neuropeptide Y GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
257010
Protein
NPY1R
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
Y2 Human Neuropeptide Y GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
257110
Protein
Y2
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
NT1 Human Neurotensin GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
258010
Protein
NT1
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
nAChR (alpha1) Human Ion Channel Binding Antagonist Radioligand LeadHunter Assay - TW
Item
258700
Protein
nAChR-a1
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
nAChR (alpha3/beta4) Human Ion Channel Binding Agonist Radioligand LeadHunter Assay - TW
Item
258730
Protein
nAChR-a3b4
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
delta (DOP) Human Opioid GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
260130
Protein
delta (DOP)
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
kappa (KOP) Human Opioid GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
260210
Protein
kappa (KOP)
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
mu (MOP) Human Opioid GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
260410
Protein
mu (MOP)
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
NOP (ORL1) Human Opioid GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
260600
Protein
NOP (ORL1)
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
OT Human Vasopressin / Oxytocin GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
260900
Protein
OT
Organism
Human
Assay Sub Type
Binding
Family
Other
Name
Phorbol Ester Binding LeadHunter Assay - TW
Item
264500
Protein
Organism
Mouse
Assay Sub Type
Binding
Family
Kinase
Name
PDGFR (Non-Selective) Mouse RTK Kinase Binding Agonist Radioligand LeadHunter Assay - TW
Item
265200
Protein
Organism
Mouse
Assay Sub Type
Binding
Family
Ion Channel
Name
KATP Hamster Potassium Ion Channel Binding Antagonist Radioligand LeadHunter Assay - TW
Item
265600
Protein
KATP
Organism
Hamster
Assay Sub Type
Binding
Family
Ion Channel
Name
Kv1.1 Human Potassium Channel Binding Antagonist Radioligand LeadHunter Assay – TW
Item
265710
Protein
Kv1.1
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
SKCa (Non-Selective) Rat Potassium Ion Channel [125I] Apamin Binding LeadHunter Assay - TW
Item
265800
Protein
Organism
Rat
Assay Sub Type
Binding
Family
Ion Channel
Name
hERG Human Potassium Ion Channel [3H] Dofetilide Binding Antagonist Radioligand LeadHunter Assay - TW
Item
265910
Protein
hERG
Organism
Human
Assay Sub Type
Binding
Family
NHR
Name
PPARgamma Human NHR Binding Agonist Radioligand LeadHunter Assay - TW
Item
267500
Protein
PPARgamma
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
DP2 Human Prostanoid GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
268030
Protein
DP2
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
DP1 Human Prostanoid GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
268060
Protein
DP1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
EP1 Human Prostanoid GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
268110
Protein
EP1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
EP2 Human Prostanoid GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
268200
Protein
EP2
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
EP4 Human Prostanoid GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
268420
Protein
EP4
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
FP Human Prostanoid GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
268510
Protein
FP
Organism
Human
Assay Sub Type
Binding
Family
NHR
Name
RARalpha Human Retinoic Acid NHR Binding (Agonist Radioligand) Assay, Panlabs
Item
269200
Protein
RARalpha
Organism
Human
Assay Sub Type
Binding
Family
NHR
Name
RXRalpha Human Retinoid X NHR Binding (Agonist Radioligand) Assay, Panlabs
Item
269500
Protein
RXRalpha
Organism
Human
Assay Sub Type
Binding
Family
PDE
Name
PDE (Non-Selective) Rat [3H] Rolipram Binding Antagonist Radioligand LeadHunter Assay - TW
Item
270000
Protein
Organism
Rat
Assay Sub Type
Binding
Family
Ion Channel
Name
RY3 Rat Ryanodine Ion Channel Binding Agonist Radioligand LeadHunter Assay - TW
Item
270300
Protein
RY3
Organism
Rat
Assay Sub Type
Binding
Family
GPCR
Name
5-HT1A Human Serotonin GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
271110
Protein
5-HT1A
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
5-HT1B Human Serotonin GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
271230
Protein
5-HT1B
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
5-HT2A Human Serotonin GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
271650
Protein
5-HT2A
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
5-HT2B Human Serotonin GPCR [3H] LSD Binding Agonist Radioligand LeadHunter Assay - TW
Item
271700
Protein
5-HT2B
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
5-HT2C Human Serotonin GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
271800
Protein
5-HT2C
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
5-HT3 Human Serotonin Ion Channel Binding Antagonist Radioligand LeadHunter Assay - TW
Item
271910
Protein
5-HT3A
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
5-HT4B Human Serotonin GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
272010
Protein
5-HT4 (B)
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
5-HT5A Human Serotonin GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
272100
Protein
5-HT5A
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
5-HT6 Human Serotonin GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
272200
Protein
5-HT6
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
5-HT7 Human Serotonin GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
272320
Protein
5-HT7
Organism
Human
Assay Sub Type
Binding
Family
Transporter
Name
SERT Human Serotonin Transporter Binding Antagonist Radioligand LeadHunter Assay - TW
Item
274030
Protein
SERT
Organism
Human
Assay Sub Type
Binding
Family
Transmembrane (Other)
Name
sigma2 Rat [3H] Ifenprodil Binding Agonist Radioligand LeadHunter Assay - TW
Item
278200
Protein
Organism
Rat
Assay Sub Type
Binding
Family
Ion Channel
Name
Nav1.5 Sodium Channel Human Ion Channel [3H]BNZA Binding LeadHunter Assay - TW
Item
279520
Protein
Nav1.5
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
sst1 Human Somatostatin GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
282510
Protein
sst1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
sst3 Human Somatostatin GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
282530
Protein
sst3
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
sst2 Human Somatostatin GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
282700
Protein
sst2
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
sst4 Human Somatostatin GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
282910
Protein
sst4
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
sst5 Human Somatostatin GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
283010
Protein
sst5
Organism
Human
Assay Sub Type
Binding
Family
NHR
Name
TR (Non-Selective) Rat Thyroid Hormone NHR Binding Agonist Radioligand LeadHunter Assay - TW
Item
285900
Protein
Organism
Rat
Assay Sub Type
Binding
Family
GPCR
Name
TRH Human Thyrotropin-RH GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
286010
Protein
TRH
Organism
Human
Assay Sub Type
Binding
Family
Kinase
Name
TGFbeta (Non-Selective) Mouse TKL Kinase Binding Agonist Radioligand LeadHunter Assay - TW
Item
286200
Protein
Organism
Mouse
Assay Sub Type
Binding
Family
GPCR
Name
UT (GPR14) Human Urotensin GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
286700
Protein
UT (GPR14)
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
VIP1 (VPAC1) Human VIP and PACAP GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
287010
Protein
VIP1 (VPAC1)
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
VIP2 (VPAC2) Human VIP and PACAP GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
287100
Protein
VIP2 (VPAC2)
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
V1A Human Vasopressin / Oxytocin GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
287530
Protein
V1A
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
V1B Human Vasopressin / Oxytocin GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
287560
Protein
V1B
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
V2 Human Vasopressin / Oxytocin GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
287610
Protein
V2
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
OX2 Human Orexin GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
299002
Protein
OX2
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
IP Human Prostanoid GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
299004
Protein
IP
Organism
Human
Assay Sub Type
Binding
Family
NHR
Name
PR Human Progesterone NHR Binding Agonist Radioligand LeadHunter Assay - TW
Item
299005
Protein
PR
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
EP3 Human Prostanoid GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
299006
Protein
EP3
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
OX1 Human Orexin GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
299030
Protein
OX1
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
nAChR (alpha4/beta2) Human Ion Channel Binding Agonist Radioligand LeadHunter Assay - TW
Item
299031
Protein
nAChR-a4b2
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
nAChR (alpha7) Human Ion Channel Binding Antagonist Radioligand LeadHunter Assay - TW
Item
299032
Protein
nAChR
Organism
Human
Assay Sub Type
Binding
Family
Transmembrane (Other)
Name
sigma1 Human Binding Agonist Radioligand LeadHunter Assay - TW
Item
299034
Protein
sigma1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
H4 Human Histamine GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
299035
Protein
H4R
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
P2X (Non-Selective) Rat Ion Channel Binding Agonist Radioligand LeadHunter Assay - TW
Item
299036
Protein
Organism
Rat
Assay Sub Type
Binding
Family
GPCR
Name
PAF Human Platelet-Activating Factor GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
299037
Protein
PAF
Organism
Human
Assay Sub Type
Binding
Assay Information
Assay Type:
Biochemical
Testing Information
Test Concentration / Dose:
Suggested concentration for initial testing is 10 µM
Test Sample Requirements:
200 μl of a 10 mM stock or 1.5 mg pre-weighed powder (assuming FW≦500 and purity 100%)
Turnaround Time
Standard:
10 Business Days
Service Scheduling Note:
SpectrumScreen Panel is initiated and run on every Thursday. Please send us the compounds and compound submission form (CSF) before 12 pm (GMT+8) Wednesday (cut-off date), to smooth the process.
Additional Information
Brand:
SafetyScreen
Testing Location:
Taiwan - Taipei
Questions? Contact Us
You can easily get in touch with a Eurofins Discovery Expert or get help from our Customer Service team. Reach out with questions, or to discuss your specific discovery challenges.
