OVERVIEW
DOCUMENTS/REFERENCES
Biological Information
No. of Assays on Panel:
67
Assays on Panel:
Family
GPCR
Name
A1 Human Adenosine GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
200510
Protein
A1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
A2A Human Adenosine GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
200610
Protein
A2A
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
A3 Human Adenosine GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
200720
Protein
A3
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
alpha1A Human Adrenoceptor GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
203110
Protein
alpha1A
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
alpha1B Human Adrenoceptor GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
203210
Protein
alpha1B
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
alpha1D Human Adrenoceptor GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
203400
Protein
alpha1D
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
alpha2A Human Adrenoceptor GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
203630
Protein
alpha2A
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
beta1 Human Adrenoceptor GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
204010
Protein
beta1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
beta2 Human Adrenoceptor GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
204110
Protein
beta2
Organism
Human
Assay Sub Type
Binding
Family
Transporter
Name
NET Human Norepinephrine Transporter Binding Antagonist Radioligand LeadHunter Assay - TW
Item
204410
Protein
NET
Organism
Human
Assay Sub Type
Binding
Family
NHR
Name
AR Human Androgen NHR Binding Agonist Radioligand LeadHunter Assay - TW
Item
206000
Protein
AR
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
B1 Human Bradykinin GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
212520
Protein
B1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
B2 Human Bradykinin GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
212620
Protein
B2
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
Cav1.2 (L-type) Rat Calcium Ion Channel Binding (Diltiazem Site) LeadHunter Assay - TW
Item
214510
Protein
Cav1.2 (L-type)
Organism
Rat
Assay Sub Type
Binding
Family
Ion Channel
Name
Cav1.2 (L-type) Human Calcium Ion Channel Binding (Dihydropyridine Site) LeadHunter Assay - TW
Item
214610
Protein
Cav1.2 (L-type)
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
Cav2.2 (N-type) Rat Calcium Ion Channel Binding Antagonist Radioligand LeadHunter Assay - TW
Item
216000
Protein
Cav2.2 (N-type)
Organism
Rat
Assay Sub Type
Binding
Family
GPCR
Name
CB1 Human Cannabinoid GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
217050
Protein
CB1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
D1 Human Dopamine GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
219500
Protein
D1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
D2S Human Dopamine GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
219700
Protein
D2
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
D3 Human Dopamine GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
219800
Protein
D3
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
D4.4 Human Dopamine GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
220000
Protein
D4
Organism
Human
Assay Sub Type
Binding
Family
Transporter
Name
DAT Human Dopamine Transporter Binding Antagonist Radioligand LeadHunter Assay - TW
Item
220320
Protein
DAT
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
ETA Human Endothelin GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
224010
Protein
ETA
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
ETB Human Endothelin GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
224110
Protein
ETB
Organism
Human
Assay Sub Type
Binding
Family
Kinase
Name
EGFR Human RTK Kinase Binding Radiometric LeadHunter Assay [10 uM ] - TW
Item
225510
Protein
EGFR
Organism
Human
Assay Sub Type
Binding
Family
NHR
Name
ERalpha Human Estrogen NHR Binding Agonist Radioligand LeadHunter Assay - TW
Item
226010
Protein
ERalpha
Organism
Human
Assay Sub Type
Binding
Family
Transporter
Name
GABA (Non-Selective) Rat Transporter Binding Antagonist Radioligand LeadHunter Assay - TW
Item
226400
Protein
Organism
Rat
Assay Sub Type
Binding
Family
Ion Channel
Name
GABAA (Non-Selective) Rat Ion Channel [3H] Muscimol Binding Agonist Radioligand LeadHunter Assay - TW
Item
226500
Protein
Organism
Rat
Assay Sub Type
Binding
Family
Ion Channel
Name
GABAA (Non-Selective) Rat Ion Channel [3H] Flunitrazepam Binding Agonist Radioligand LeadHunter Assay - TW
Item
226600
Protein
Organism
Rat
Assay Sub Type
Binding
Family
GPCR
Name
GABAB (B1a/B2) Human GABAB GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
228610
Protein
GABAB (B1/B2)
Organism
Human
Assay Sub Type
Binding
Family
NHR
Name
GR Human Glucocorticoid NHR Binding Agonist Radioligand LeadHunter Assay - TW
Item
232030
Protein
GR
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
Glutamate (Kainate, Non-Selective) Rat Ion Channel [3H] Kainic acid Binding LeadHunter Assay - TW
Item
232710
Protein
Organism
Rat
Assay Sub Type
Binding
Family
Ion Channel
Name
Glutamate (NMDA, NR1/NR2A) Human Ion Channel [3H] CGP-39653 Binding LeadHunter Assay - TW
Item
232820
Protein
GluN1/ GluN2A
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
Glutamate (NMDA, Non-Selective) Rat Ion Channel [3H] MDL 105,519 Binding LeadHunter Assay - TW
Item
232910
Protein
Organism
Rat
Assay Sub Type
Binding
Family
Ion Channel
Name
Glutamate (Non-Selective) Rat Ion Channel [3H] TCP Binding LeadHunter Assay - TW
Item
233000
Protein
Organism
Rat
Assay Sub Type
Binding
Family
GPCR
Name
H1 Human Histamine GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
239610
Protein
H1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
H2 Human Histamine GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
239710
Protein
H2
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
H3 Human Histamine GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
239820
Protein
H3
Organism
Human
Assay Sub Type
Binding
Family
Transmembrane (Other)
Name
Imidazoline I2 Central Rat Binding Antagonist Radioligand LeadHunter Assay - TW
Item
241000
Protein
Organism
Rat
Assay Sub Type
Binding
Family
Cell Surface (Other)
Name
IL-1 R1 Human Interleukin Binding Agonist Radioligand LeadHunter Assay - TW
Item
243530
Protein
IL-1R-1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
CysLT1 Human Leukotriene GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
250460
Protein
CysLT1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
MT1 Human Melatonin GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
251600
Protein
MT1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
M1 Human Acetylcholine (Muscarinic) GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
252610
Protein
M1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
M2 Human Acetylcholine (Muscarinic) GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
252710
Protein
M2
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
M3 Human Acetylcholine (Muscarinic) GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
252810
Protein
M3
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
NK1 Human Tachykinin GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
255520
Protein
NK1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
Y1 Human Neuropeptide Y GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
257010
Protein
NPY1R
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
Y2 Human Neuropeptide Y GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
257110
Protein
Y2
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
nAChR (alpha1) Human Ion Channel Binding Antagonist Radioligand LeadHunter Assay - TW
Item
258700
Protein
nAChR-a1
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
nAChR (alpha3/beta4) Human Ion Channel Binding Agonist Radioligand LeadHunter Assay - TW
Item
258730
Protein
nAChR-a3b4
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
delta (DOP) Human Opioid GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
260130
Protein
delta (DOP)
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
kappa (KOP) Human Opioid GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
260210
Protein
kappa (KOP)
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
mu (MOP) Human Opioid GPCR Binding Antagonist Radioligand LeadHunter Assay - TW
Item
260410
Protein
mu (MOP)
Organism
Human
Assay Sub Type
Binding
Family
Other
Name
Phorbol Ester Binding LeadHunter Assay - TW
Item
264500
Protein
Organism
Mouse
Assay Sub Type
Binding
Family
Ion Channel
Name
KATP Hamster Potassium Ion Channel Binding Antagonist Radioligand LeadHunter Assay - TW
Item
265600
Protein
KATP
Organism
Hamster
Assay Sub Type
Binding
Family
Ion Channel
Name
hERG Human Potassium Ion Channel [3H] Dofetilide Binding Antagonist Radioligand LeadHunter Assay - TW
Item
265910
Protein
hERG
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
EP4 Human Prostanoid GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
268420
Protein
EP4
Organism
Human
Assay Sub Type
Binding
Family
PDE
Name
PDE (Non-Selective) Rat [3H] Rolipram Binding Antagonist Radioligand LeadHunter Assay - TW
Item
270000
Protein
Organism
Rat
Assay Sub Type
Binding
Family
GPCR
Name
5-HT1A Human Serotonin GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
271110
Protein
5-HT1A
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
5-HT2B Human Serotonin GPCR [3H] LSD Binding Agonist Radioligand LeadHunter Assay - TW
Item
271700
Protein
5-HT2B
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
5-HT3 Human Serotonin Ion Channel Binding Antagonist Radioligand LeadHunter Assay - TW
Item
271910
Protein
5-HT3A
Organism
Human
Assay Sub Type
Binding
Family
Transporter
Name
SERT Human Serotonin Transporter Binding Antagonist Radioligand LeadHunter Assay - TW
Item
274030
Protein
SERT
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
Nav1.5 Sodium Channel Human Ion Channel [3H]BNZA Binding LeadHunter Assay - TW
Item
279520
Protein
Nav1.5
Organism
Human
Assay Sub Type
Binding
Family
NHR
Name
TR (Non-Selective) Rat Thyroid Hormone NHR Binding Agonist Radioligand LeadHunter Assay - TW
Item
285900
Protein
Organism
Rat
Assay Sub Type
Binding
Family
Transmembrane (Other)
Name
sigma1 Human Binding Agonist Radioligand LeadHunter Assay - TW
Item
299034
Protein
sigma1
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
P2X (Non-Selective) Rat Ion Channel Binding Agonist Radioligand LeadHunter Assay - TW
Item
299036
Protein
Organism
Rat
Assay Sub Type
Binding
Family
GPCR
Name
PAF Human Platelet-Activating Factor GPCR Binding Agonist Radioligand LeadHunter Assay - TW
Item
299037
Protein
PAF
Organism
Human
Assay Sub Type
Binding
Assay Information
Assay Type:
Biochemical
Assay Sub Type:
Binding
Testing Information
Test Concentration / Dose:
Suggested concentration for initial testing is 10 µM
Test Sample Requirements:
150 μl of a 10 mM stock or 1 mg pre-weighed powder (assuming FW≦500 and purity 100%)
Turnaround Time
Standard:
10 Business Days
Additional Information
Brand:
SafetyScreen
Testing Location:
Taiwan - Taipei
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