GIP Human Gastric Inhibitory Polypeptide GPCR Binding Agonist Radioligand LeadHunter assay - FR
OVERVIEW
DOCUMENTS/REFERENCES
Biological Information
Background Information:
Evaluation of the affinity of compounds for the human GIP receptor, determined in a radioligand competition binding assay.
Family:
GPCR
Sub Family:
Glucagon
Class:
Class B
Protein Name:
GIP
Uniprot Number:
P48546
Protein Aliases:
Glucose-dependent insulinotropic polypeptide receptor
Gene Name:
GIPR
Gene ID:
2696
Gene Aliases:
gastric inhibitory polypeptide receptor
Accession Number:
P48546
Organism:
Human
Assay Information
Assay Type:
Biochemical
Assay Sub Type:
Binding
Detection Method:
Radiometric
Testing Information
Ligand:
[125I]GIP
Ligand Kd (nM):
0,62
Ligand Concentration:
0,05 nM
Non Specific:
GIP(h) (1 µM)
Incubation:
2h at 22°C
Test Sample Requirements:
Minimum for 1) Screen: 60 μl of 10 mM stock -OR- 1 mg (pre-weighed) for 10µM final testing. 2) Dose Response: 90 μl of 10 mM stock -OR- 1 mg (pre-weighed) for a top concentration at 10 µM.
Minimum Order Quantity:
2
Turnaround Time
Standard:
15 Business Days
Reference Compound Data
Additional Information
Brand:
LeadHunter
Testing Location:
France - Celle L'Evescault
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