OVERVIEW
DOCUMENTS/REFERENCES
Biological Information
Background Information:
Panel of GPCR β-arrestin or second messenger assays and dimerization assay that can be used to measure specificity or selectivity during Hit to Lead or Lead Optimization stages of drug development.
No. of Assays on Panel:
25
Assays on Panel:
Family
GPCR
Name
GIP Human Glucagon GPCR Cell Based Agonist Arrestin LeadHunter Assay - US
Item
86-0001P-2059AG
Protein
GIP
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
CT Human Calcitonin GPCR Cell Based Agonist Arrestin LeadHunter Assay - US
Item
86-0001P-2114AG
Protein
CT
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
AMY3 (CT/RAMP3) Human Calcitonin GPCR Cell Based Agonist Arrestin LeadHunter Assay - US
Item
86-0001P-2116AG
Protein
CT
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
CCK1 (CCKA) Human Cholecystokinin GPCR Cell Based Agonist Arrestin LeadHunter Assay - US
Item
86-0001P-2138AG
Protein
CCK1 (CCKA)
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
GHSR Human Ghrelin GPCR Cell Based Antagonist Arrestin LeadHunter Assay - US
Item
86-0001P-2164AN
Protein
GHSR
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
Glucagon Human Glucagon GPCR Cell Based Agonist Arrestin LeadHunter Assay - US
Item
86-0001P-2165AG
Protein
Glucagon
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
GLP-1 Human Glucagon GPCR Cell Based Agonist Arrestin LeadHunter Assay - US
Item
86-0001P-2166AG
Protein
GLP-1
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
MC4 Human Melanocortin GPCR Cell Based Agonist Arrestin LeadHunter Assay - US
Item
86-0001P-2189AG
Protein
MC4
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
Y2 Human Neuropeptide Y GPCR Cell Based Agonist Arrestin LeadHunter Assay - US
Item
86-0001P-2198AG
Protein
Y2
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
Y4 Human Neuropeptide Y GPCR Cell Based Agonist Arrestin LeadHunter Assay - US
Item
86-0001P-2199AG
Protein
Y4
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
OX1 Human Orexin GPCR Cell Based Antagonist Arrestin LeadHunter Assay - US
Item
86-0001P-2205AN
Protein
OX1
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
OX2 Human Orexin GPCR Cell Based Antagonist Arrestin LeadHunter Assay - US
Item
86-0001P-2206AN
Protein
OX2
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
CT Human Calcitonin GPCR Cell Based Agonist cAMP LeadHunter Assay - US
Item
86-0007P-2245AG
Protein
CT
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
Glucagon Human Glucagon GPCR Cell Based Agonist cAMP LeadHunter Assay - US
Item
86-0007P-2306AG
Protein
Glucagon
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
GIP Human Glucagon GPCR in CHO Cell Based Agonist cAMP LeadHunter Assay - US
Item
86-0007P-2308AG
Protein
GIP
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
GLP-1 Human Glucagon GPCR Cell Based Agonist cAMP LeadHunter Assay - US
Item
86-0007P-2309AG
Protein
GLP-1
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
MC4 Human Melanocortin GPCR Cell Based Agonist cAMP LeadHunter Assay - US
Item
86-0007P-2326AG
Protein
MC4
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
Y2 Human Neuropeptide Y GPCR Cell Based Agonist cAMP LeadHunter Assay - US
Item
86-0007P-2337AG
Protein
Y2
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
Y4 Human Neuropeptide Y GPCR Cell Based Agonist cAMP LeadHunter Assay - US
Item
86-0007P-2338AG
Protein
Y4
Organism
Human
Assay Sub Type
Cell Based
Family
Cell Surface (Other)
Name
LEPR/LEPR Human Cytokine Cell Based Agonist Dimerization LeadHunter Assay - US
Item
86-0020P-2661AG
Protein
LEPR
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
CCK1 (CCKA) Human Cholecystokinin GPCR Cell Based Agonist Calcium Flux (in Arrestin Cell Line) LeadHunter Assay - US
Item
86-0030P-2138AG
Protein
CCK1 (CCKA)
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
GHSR Human Ghrelin GPCR Cell Based Antagonist Calcium Flux (in Arrestin Cell Line) LeadHunter Assay - US
Item
86-0030P-2164AN
Protein
GHSR
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
OX1 Human Orexin GPCR Cell Based Antagonist Calcium Flux (in Arrestin Cell Line) LeadHunter Assay - US
Item
86-0030P-2205AN
Protein
OX1
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
OX2 Human Orexin GPCR Cell Based Antagonist Calcium Flux (in Arrestin Cell Line) LeadHunter Assay - US
Item
86-0030P-2206AN
Protein
OX2
Organism
Human
Assay Sub Type
Cell Based
Family
GPCR
Name
AMY3 (CT/RAMP3) Human Calcitonin GPCR Cell Based Agonist cAMP (TR-FRET in Arrestin Cell Line) LeadHunter Assay - US
Item
86-3002P-2276AG
Protein
CT
Organism
Human
Assay Sub Type
Cell Based
Family:
GPCR
Organism:
Human
Assay Information
Assay Type:
Functional
Assay Sub Type:
Cell Based
Testing Information
Test Sample Requirements:
75uL of a 1000X stock based on the final concentration being tested
Turnaround Time
Standard:
20 Business Days
Service Scheduling Note:
Turnaround time is twenty-two (22) business days from the project initiation.
Additional Information
Brand:
DiscoverX
Testing Location:
USA - Fremont, CA
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