OVERVIEW
DOCUMENTS/REFERENCES
Biological Information
Background Information:
Delta SafetyScreen87 - SafetyScreen44 Panel. Only to consider if you already run a Safetyscreen44 with us.
No. of Assays on Panel:
43
Assays on Panel:
Family
GPCR
Name
NK1 Human Tachykinin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
100
Protein
NK1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
Y1 Human Neuropeptide Y GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
106
Protein
Y1
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
Glutamate (Non-Selective) Rat Ion Channel [3H] TCP Binding LeadHunter Assay - FR
Item
124
Protein
NMDA(PCP site)
Organism
Rat
Assay Sub Type
Binding
Family
GPCR
Name
alpha2B Human Adrenoceptor GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
1344
Protein
alpha2B
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
5-HT2C Human Serotonin GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
137
Protein
5-HT2C
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
D2L Human Dopamine GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
1405
Protein
D2
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
Cav1.2 (L-type) Rat Calcium Ion Channel Binding (Verapamil Site) LeadHunter Assay - FR
Item
163
Protein
CaV1.2 (Vera. site)
Organism
Rat
Assay Sub Type
Binding
Family
GPCR
Name
alpha1B Human Adrenoceptor GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
1633
Protein
alpha1B
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
Cav2.2 (N-type) Rat Calcium Ion Channel Binding Antagonist Radioligand LeadHunter Assay - FR
Item
164
Protein
Cav2.2 (N-type)
Organism
Rat
Assay Sub Type
Binding
Family
Protease
Name
Cathepsin G Human Chymotrypsin Serine Peptidase Enzymatic LeadHunter Assay - FR
Item
179
Protein
Cathepsin G
Organism
Human
Assay Sub Type
Enzymatic
Family
GPCR
Name
alpha1D Human Adrenoceptor GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
1942
Protein
alpha1D
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
A1 Human Adenosine GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
2
Protein
A1
Organism
Human
Assay Sub Type
Binding
Family
Transporter
Name
ATPase (Na+/K+) Pig Brain Enzymatic LeadHunter Assay - FR
Item
2009
Protein
Na/K ATPase
Organism
Pig
Assay Sub Type
Enzymatic
Family
NHR
Name
RARalpha Human Retinoic Acid NHR Binding Agonist Radioligand LeadHunter Assay - FR
Item
2084
Protein
RARalpha
Organism
Human
Assay Sub Type
Binding
Family
NHR
Name
PR Human Progesterone NHR Binding Agonist Radioligand LeadHunter Assay - FR
Item
2341
Protein
PR
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
AT1 Human Angiotensin GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
24
Protein
AT1
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
GABAA (alpha1/beta2/gamma2) Human Ion Channel [3H] Muscimol Binding Agonist Radioligand LeadHunter Assay - FR
Item
3051
Protein
GABAA
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
B2 Human Bradykinin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
33
Protein
B2
Organism
Human
Assay Sub Type
Binding
Family
Protease
Name
ACE Human Angiotensin-Converting Metallo Peptidase Enzymatic LeadHunter Assay - FR
Item
3441
Protein
ACE
Organism
Human
Assay Sub Type
Enzymatic
Family
Enzyme
Name
Monoamine Oxidase B (MAO-B) Human Enzymatic LeadHunter Assay - FR
Item
3477
Protein
MAO-B
Organism
Human
Assay Sub Type
Enzymatic
Family
GPCR
Name
CCR1 Human Chemokine GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
361
Protein
CCR1
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
GABAA (Non-Selective) Rat Ion Channel [3H] TBOB Binding Antagonist Radioligand LeadHunter Assay - FR
Item
3817
Protein
GABAA (TBOB site)
Organism
Rat
Assay Sub Type
Binding
Family
GPCR
Name
mGlu5 Human Glutamate (Metabotropic) GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
3844
Protein
mGlu5
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
CCK2 (CCKB) Human Cholecystokinin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
41
Protein
CCK2 (CCKB)
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
CXCR2 (IL-8RB) Human Chemokine GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
419
Protein
CXCR2 (IL-8RB)
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
MC4 Human Melanocortin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
420
Protein
MC4
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
Cav1.2 (L-type) Human Calcium Ion Channel Binding (diltiazem site) (benzothiazepines) LeadHunter Assay - FR
Item
4549
Protein
Cav1.2 (L-type)
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
PAF Human Platelet-Activating Factor GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
4569
Protein
PAF
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
GABAB (B1b/B2) Human GABAB GPCR Mass Spectrometry Binding Antagonist ligand LeadHunter Assay - FR
Item
4699
Protein
GABAB (B1/B2)
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
Glutamate (Non-Selective) Rat Ion Channel Glycine (Strychnine-Insensitive) Mass Spectrometry Binding LeadHunter Assay - FR
Item
5043
Protein
NMDA(strychine-insensitive site)
Organism
Rat
Assay Sub Type
Binding
Family
Ion Channel
Name
Glycine (Non-Selective) Rat Ion Channel Strychnine Mass Spectrometry Binding LeadHunter Assay - FR
Item
5044
Protein
alpha-1 GlyR
Organism
Rat
Assay Sub Type
Binding
Family
Transporter
Name
Adenosine Guinea Pig Transporter Mass Spectrometry Binding Antagonist Ligand LeadHunter Assay - FR
Item
5113
Protein
SLC29A1
Organism
Guinea Pig
Assay Sub Type
Binding
Family
Ion Channel
Name
GluK2 Human Ion Channel [3H] Kainic acid Binding LeadHunter Assay - FR
Item
5379
Protein
Kainate
Organism
Human
Assay Sub Type
Binding
Family
NHR
Name
ERalpha Human Estrogen NHR Binding Agonist Radioligand LeadHunter Assay - FR
Item
5484
Protein
ERalpha
Organism
Human
Assay Sub Type
Binding
Family
Kinase
Name
IR (INSR) Human RTK Kinase Enzymatic Radiometric [Km ATP] SafetyScreen - FR
Item
5623
Protein
IR
Organism
Human
Assay Sub Type
Enzymatic
Family
Kinase
Name
PKCalpha Human PKC Kinase Enzymatic Radiometric [Km ATP] SafetyScreen - FR
Item
5625
Protein
PKCalpha
Organism
Human
Assay Sub Type
Enzymatic
Family
Transporter
Name
GAT1 Human GABA Transporter Binding Antagonist Radioligand LeadHunter Assay - FR
Item
5773
Protein
GAT-1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
CysLT1 Human Leukotriene GPCR Mass Spectrometry Binding Agonist ligand LeadHunter Assay - FR
Item
5841
Protein
CYSLT1
Organism
Human
Assay Sub Type
Binding
Family
Ion Channel
Name
Glutamate (AMPA, Non-Selective) Rat Ion Channel [3H] AMPA Binding LeadHunter Assay - FR
Item
64
Protein
AMPA
Organism
Rat
Assay Sub Type
Binding
Family
NHR
Name
PPARgamma Human NHR Binding Agonist Radioligand LeadHunter Assay - FR
Item
641
Protein
PPARgamma
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
MC1 Mouse Melanocortin GPCR Binding Agonist Radioligand LeadHunter Assay - FR
Item
644
Protein
MC1
Organism
Mouse
Assay Sub Type
Binding
Family
Ion Channel
Name
nAChR (Alpha1, Muscle-Type) Human Ion Channel Binding Antagonist Radioligand LeadHunter Assay - FR
Item
936
Protein
nAChR-α1
Organism
Human
Assay Sub Type
Binding
Family
GPCR
Name
M4 Human Acetylcholine (Muscarinic) GPCR Binding Antagonist Radioligand LeadHunter Assay - FR
Item
96
Protein
M4
Organism
Human
Assay Sub Type
Binding
Testing Information
Test Sample Requirements:
Minimum for Screen: 120 μl of 10 mM stock -OR- 1 mg (pre-weighed) for 10µM final testing.
(PBS or HBSS working solutions are not compatible)
Turnaround Time
Standard:
10 Business Days
Additional Information
Brand:
SafetyScreen
Testing Location:
France - Celle L'Evescault
RELATED SOLUTIONS
SafetyScreen44 Panel - FR
Item: P270
SafetyScreen87 Panel - FR
Item: P342
SafetyScreen Functional Panel - FR
Item: P347
SafetyScreen18 Core Panel - FR
Item: P447
SafetyScreen59 Extended Panel - FR
Item: P448
SafetyScreen33 Delta Panel - FR
Item: P453
SafetyScreen Kinase Panel [1mM ATP] - FR
Item: P454
SafetyScreen77 Core Extended Panel - FR
Item: P456
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